Literature DB >> 15664824

Acyl sulfonamide anti-proliferatives. Part 2: activity of heterocyclic sulfonamide derivatives.

Mary M Mader1, Chuan Shih, Eileen Considine, Alfonso De Dios, Cora Sue Grossman, Philip A Hipskind, Ho-Shen Lin, Karen L Lobb, Beatriz Lopez, José E Lopez, Luisa M Martin Cabrejas, Michael E Richett, Wesley T White, Yiu-Yin Cheung, Zhongping Huang, John E Reilly, Sean R Dinn.   

Abstract

The anti-proliferative activity of acylated heterocyclic sulfonamides is described in Vascular Endothelial Growth Factor-dependent Human Umbilical Vascular Endothelial Cells (VEGF-HUVEC) and in HCT116 tumor cells in a soft agar diffusion assay.

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Year:  2005        PMID： 15664824     DOI： 10.1016/j.bmcl.2004.11.041

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

1.  Iridium-Catalyzed Silylation of Five-Membered Heteroarenes: High Sterically Derived Selectivity from a Pyridyl-Imidazoline Ligand.

Authors:  Caleb Karmel; Camille Z Rubel; Elena V Kharitonova; John F Hartwig
Journal:  Angew Chem Weinheim Bergstr Ger       Date:  2020-01-22

2.  A p-methoxybenzyl (PMB) protection/deprotection approach toward the synthesis of 5-phenoxy-4-chloro-N-(aryl/alkyl) thiophene-2-sulfonamides.

Authors:  Alfred L Williams; Srinivasa R Dandepally; Sharadsrikar V Kotturi
Journal:  Mol Divers       Date:  2009-11-21       Impact factor: 2.943

3.  Crystal structures of isomeric 4-bromo-N-[(2-nitro-phen-yl)sulfon-yl]benzamide and 4-bromo-N-[(4-nitro-phen-yl)sulfon-yl]benzamide.

Authors:  S Naveen; A G Sudha; E Suresha; N K Lokanath; P A Suchetan; M Abdoh
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2017-02-03

4.  An insight into the pharmacophores of phosphodiesterase-5 inhibitors from synthetic and crystal structural studies.

Authors:  Gong Chen; Huanchen Wang; Howard Robinson; Jiwen Cai; Yiqian Wan; Hengming Ke
Journal:  Biochem Pharmacol       Date:  2008-02-12       Impact factor: 5.858

5.  Crystal structures of three N-(aryl-sulfon-yl)-4-fluoro-benzamides.

Authors:  P A Suchetan; S Naveen; N K Lokanath; K S Srivishnu; G M Supriya; H N Lakshmikantha
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2016-03-31

6.  Crystal structures of N-(3-fluoro-benzo-yl)benzene-sulfonamide and N-(3-fluoro-benzo-yl)-4-methyl-benzene-sulfonamide.

Authors:  P A Suchetan; S Naveen; N K Lokanath; H N Lakshmikantha; K S Srivishnu; G M Supriya
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2016-03-02
  6 in total

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