Literature DB >> 15651803

Investigations of the halogen dance reaction on N-substituted 2-thiazolamines.

Peter Stanetty1, Michael Schnürch, Kurt Mereiter, Marko D Mihovilovic.   

Abstract

The halogen dance (HD) reaction on various 2-thiazolamine systems was investigated providing an easy access to a series of 5-substituted 4-bromo-2-thiazolamine derivatives. We could show that HD is a very favored process for the investigated systems and that prevention of HD is only possible when optimized reaction conditions and selected electrophiles are applied.

Entities:  

Year:  2005        PMID： 15651803     DOI： 10.1021/jo0484326

Source DB:  PubMed          Journal:  J Org Chem        ISSN： 0022-3263            Impact factor:   4.354


  4 in total

1.  Methodology for the Synthesis of Substituted 1,3-Oxazoles.

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Journal:  Synlett       Date:  2009-12-22       Impact factor: 2.454

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Journal:  ChemMedChem       Date:  2021-10-22       Impact factor: 3.466

3.  Organolithium-Mediated Postfunctionalization of Thiazolo[3,2-c][1,3,5,2]oxadiazaborinine Fluorescent Dyes.

Authors:  Mykhaylo A Potopnyk; Dmytro Volyniuk; Roman Luboradzki; Magdalena Ceborska; Iryna Hladka; Yan Danyliv; Juozas V Grazulevicius
Journal:  J Org Chem       Date:  2020-04-21       Impact factor: 4.354

4.  Structure-activity relationship studies in substituted sulfamoyl benzamidothiazoles that prolong NF-κB activation.

Authors:  Nikunj M Shukla; Michael Chan; Fitzgerald S Lao; Paul J Chu; Masiel Belsuzarri; Shiyin Yao; Jason Nan; Fumi Sato-Kaneko; Tetsuya Saito; Tomoko Hayashi; Maripat Corr; Dennis A Carson; Howard B Cottam
Journal:  Bioorg Med Chem       Date:  2021-05-30       Impact factor: 3.641
  4 in total

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