Literature DB >> 15602603

Application of tandem Ugi multi-component reaction/ring closing metathesis to the synthesis of a conformationally restricted cyclic pentapeptide.

Silvia Anthoine Dietrich1, Luca Banfi, Andrea Basso, Gianluca Damonte, Giuseppe Guanti, Renata Riva.   

Abstract

A conformationally restricted cyclic pentapeptide, containing an unsaturated 9-membered lactam as a semi-rigid scaffold, was prepared in a very convergent manner, through tandem Ugi reaction/ring closing metathesis.

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Year:  2004        PMID: 15602603     DOI: 10.1039/b414374d

Source DB:  PubMed          Journal:  Org Biomol Chem        ISSN: 1477-0520            Impact factor:   3.876


  2 in total

Review 1.  Isocyanide-based multicomponent reactions towards cyclic constrained peptidomimetics.

Authors:  Gijs Koopmanschap; Eelco Ruijter; Romano Va Orru
Journal:  Beilstein J Org Chem       Date:  2014-03-04       Impact factor: 2.883

2.  Sulfur-Switch Ugi Reaction for Macrocyclic Disulfide-Bridged Peptidomimetics.

Authors:  Thimmalapura M Vishwanatha; Enrico Bergamaschi; Alexander Dömling
Journal:  Org Lett       Date:  2017-06-05       Impact factor: 6.005

  2 in total

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