Literature DB >> 15553227

Influence of spinline stress on release properties of a coaxial controlled release device based on EVA polymers.

Hans van Laarhoven1, Jan Veurink, Marc-Anton Kruft, Herman Vromans.   

Abstract

PURPOSE: To investigate the influence of the extrusion parameters on the polymeric structure and release properties of polyethylene vinyl acetate (EVA) coaxial fibers, used for controlled release of steroids.
METHODS: Coaxial fibers were prepared under various extrusion conditions. Both spinline stress and release properties were determined. The polymeric structure of the membrane was investigated with wide angle X-ray scattering (WAXS).
RESULTS: Upon leaving the spinneret, the polymeric fiber exhibits a large die swell. As a consequence, it is necessary to apply a force to draw the fiber to its desired diameter. A larger drawing force is needed at lower extrusion temperature, at a smaller air gap, or at a higher spinning velocity. It was found that the release rate of a steroid from the coaxial fiber increases, when the fibers are prepared at a higher spinline stress. X-ray measurements reveal that at higher spinline stress, the crystalline volume fraction of the membrane decreases. As a result of a decreasing crystallinity, the permeability of the polymer increases.
CONCLUSIONS: It is demonstrated that the extrusion parameters and spinline stress have a significant influence on the polymeric structure of the membrane and hence the release properties. Higher spinline stress results in a higher release rate.

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Year:  2004        PMID: 15553227     DOI: 10.1023/b:pham.0000045234.70538.29

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  1 in total

1.  In vitro release properties of etonogestrel and ethinyl estradiol from a contraceptive vaginal ring.

Authors:  J A H van Laarhoven; M A B Kruft; H Vromans
Journal:  Int J Pharm       Date:  2002-01-31       Impact factor: 5.875

  1 in total
  3 in total

Review 1.  Twin-screw extrusion of sustained-release oral dosage forms and medical implants.

Authors:  Xin Feng; Feng Zhang
Journal:  Drug Deliv Transl Res       Date:  2018-12       Impact factor: 4.617

2.  Dissolution from Ethylene Vinyl Acetate Copolymer Long-Acting Implants: Effect of Model Active Ingredient Size and Shape.

Authors:  Anne M Gohn; Amy Nolte; Ethan Ravotti; Seth P Forster; Morgan Giles; Nathan Rudd; Gamini Mendis
Journal:  Pharmaceutics       Date:  2022-05-27       Impact factor: 6.525

Review 3.  In Vitro Methods for Evaluating Drug Release of Vaginal Ring Formulations-A Critical Review.

Authors:  Katharina Tietz; Sandra Klein
Journal:  Pharmaceutics       Date:  2019-10-16       Impact factor: 6.321

  3 in total

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