Literature DB >> 15496058

One-pot synthesis of 1,4-disubstituted 1,2,3-triazoles from in situ generated azides.

Alina K Feldman1, Benoît Colasson, Valery V Fokin.   

Abstract

[reaction: see text] 1,4-Disubstituted 1,2,3-triazoles are obtained in excellent yields by a convenient one-pot procedure from a variety of readily available aromatic and aliphatic halides without isolation of potentially unstable organic azide intermediates.

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Year:  2004        PMID： 15496058     DOI： 10.1021/ol048859z

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  22 in total

1.  Catalytic stereoselective synthesis of diverse oxindoles and spirooxindoles from isatins.

Authors:  Jacob P MacDonald; Joseph J Badillo; Gary E Arevalo; Abel Silva-García; Annaliese K Franz
Journal:  ACS Comb Sci       Date:  2012-04-02       Impact factor: 3.784

2.  Fast dye salts provide fast access to azidoarene synthons in multi-step one-pot tandem click transformations.

Authors:  James T Fletcher; Jacquelline E Reilly
Journal:  Tetrahedron Lett       Date:  2011-10-19       Impact factor: 2.415

3.  Synthesis of C-glycosyl-bis-1,2,3-triazole derivatives from 3,4,6-tri-O-acetyl-D-glucal.

Authors:  Anwar Shamim; Frederico B Souza; Gustavo H G Trossini; Fernando M Gatti; Hélio A Stefani
Journal:  Mol Divers       Date:  2015-01-14       Impact factor: 2.943

4.  The Davis-Beirut reaction: N1,N2-disubstituted-1H-indazolones via 1,6-electrophilic addition to 3-alkoxy-2H-indazoles.

Authors:  Wayne E Conrad; Ryo Fukazawa; Makhluf J Haddadin; Mark J Kurth
Journal:  Org Lett       Date:  2011-05-25       Impact factor: 6.005

5.  2-triazole-substituted adenosines: a new class of selective A3 adenosine receptor agonists, partial agonists, and antagonists.

Authors:  Liesbet Cosyn; Krishnan K Palaniappan; Soo-Kyung Kim; Heng T Duong; Zhan-Guo Gao; Kenneth A Jacobson; Serge Van Calenbergh
Journal:  J Med Chem       Date:  2006-12-14       Impact factor: 7.446

Review 6.  Copper-catalyzed azide-alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(I) acetylides.

Authors:  Jason E Hein; Valery V Fokin
Journal:  Chem Soc Rev       Date:  2010-03-04       Impact factor: 54.564

7.  Facile Quenching and Spatial Patterning of Cylooctynes via Strain-Promoted Alkyne-Azide Cycloaddition of Inorganic Azides.

Authors:  Matthew Bjerknes; Hazel Cheng; Christopher D McNitt; Vladimir V Popik
Journal:  Bioconjug Chem       Date:  2017-05-09       Impact factor: 4.774

8.  Synthesis, characterization, and NMR studies of 1,2,3-triazolium ionic liquids: a good perspective regarding cytotoxicity.

Authors:  Nicolas Glanzmann; Arturene M L Carmo; Luciana M R Antinarelli; Elaine S Coimbra; Luiz Antônio S Costa; Adilson D da Silva
Journal:  J Mol Model       Date:  2018-06-14       Impact factor: 1.810

9.  Synthesis and anti-cancer screening of novel heterocyclic-(2H)-1,2,3-triazoles as potential anti-cancer agents.

Authors:  Narsimha Reddy Penthala; Leena Madhukuri; Shraddha Thakkar; Nikhil Reddy Madadi; Gauri Lamture; Robert L Eoff; Peter A Crooks
Journal:  Medchemcomm       Date:  2015-06-30       Impact factor: 3.597

10.  Quick assembly of 1,4-diphenyltriazoles as probes targeting beta-amyloid aggregates in Alzheimer's disease.

Authors:  Wenchao Qu; Mei-Ping Kung; Catherine Hou; Shunichi Oya; Hank F Kung
Journal:  J Med Chem       Date:  2007-06-15       Impact factor: 7.446
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