Literature DB >> 15293980

Peroxisome proliferator-activated receptor alpha/gamma dual agonists for the treatment of type 2 diabetes.

Brad R Henke1.   

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Year:  2004        PMID: 15293980     DOI: 10.1021/jm030631e

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  13 in total

1.  4',6-Dimethoxyisoflavone-7-O-β-D-glucopyranoside (wistin) is a peroxisome proliferator-activated receptor α (PPARα) agonist in mouse hepatocytes.

Authors:  Misato Suzuki; Fumiya Nakamura; Emi Taguchi; Maho Nakata; Fumi Wada; Momoka Takihi; Tomoyo Inoue; Shinji Ohta; Hiroyuki Kawachi
Journal:  Mol Cell Biochem       Date:  2018-01-09       Impact factor: 3.396

Review 2.  Interrelationship between diabetes mellitus and heart failure: the role of peroxisome proliferator-activated receptors in left ventricle performance.

Authors:  Evangelos Oikonomou; Konstantinos Mourouzis; Petros Fountoulakis; Georgios Angelos Papamikroulis; Gerasimos Siasos; Alexis Antonopoulos; Georgia Vogiatzi; Sotiris Tsalamadris; Manolis Vavuranakis; Dimitris Tousoulis
Journal:  Heart Fail Rev       Date:  2018-05       Impact factor: 4.214

3.  The peroxisome proliferator-activated receptor-gamma agonist pioglitazone represses inflammation in a peroxisome proliferator-activated receptor-alpha-dependent manner in vitro and in vivo in mice.

Authors:  Gabriela Orasanu; Ouliana Ziouzenkova; Pallavi R Devchand; Vedika Nehra; Osama Hamdy; Edward S Horton; Jorge Plutzky
Journal:  J Am Coll Cardiol       Date:  2008-07-02       Impact factor: 24.094

4.  Synthesis of tryptoline-3-carboxylic Acid derivatives a novel antidiabetic agent.

Authors:  An Choudhary; Ms Kohli; A Kumar; A Joshi
Journal:  J Young Pharm       Date:  2011-04

5.  In silico profiling for secondary metabolites from Lepidium meyenii (maca) by the pharmacophore and ligand-shape-based joint approach.

Authors:  Fan Yi; Xiao-Lei Tan; Xin Yan; Hai-Bo Liu
Journal:  Chin Med       Date:  2016-09-26       Impact factor: 5.455

6.  Find novel dual-agonist drugs for treating type 2 diabetes by means of cheminformatics.

Authors:  Lei Liu; Ying Ma; Run-Ling Wang; Wei-Ren Xu; Shu-Qing Wang; Kuo-Chen Chou
Journal:  Drug Des Devel Ther       Date:  2013-04-08       Impact factor: 4.162

7.  PPAR-gamma, Microglial Cells, and Ocular Inflammation: New Venues for Potential Therapeutic Approaches.

Authors:  Fiorella Malchiodi-Albedi; Andrea Matteucci; Antonietta Bernardo; Luisa Minghetti
Journal:  PPAR Res       Date:  2008       Impact factor: 4.964

8.  Cryptochrome and Period Proteins Are Regulated by the CLOCK/BMAL1 Gene: Crosstalk between the PPARs/RXRalpha-Regulated and CLOCK/BMAL1-Regulated Systems.

Authors:  Koh-Ichi Nakamura; Ikuo Inoue; Seiichiro Takahashi; Tsugikazu Komoda; Shigehiro Katayama
Journal:  PPAR Res       Date:  2008       Impact factor: 4.964

9.  Are fish oil omega-3 long-chain fatty acids and their derivatives peroxisome proliferator-activated receptor agonists?

Authors:  Osman A B S M Gani
Journal:  Cardiovasc Diabetol       Date:  2008-03-20       Impact factor: 9.951

Review 10.  Peroxisome proliferator-activated receptors and their ligands: nutritional and clinical implications--a review.

Authors:  Bogna Grygiel-Górniak
Journal:  Nutr J       Date:  2014-02-14       Impact factor: 3.271

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