Literature DB >> 15259086

Effect of octreotide on human pancreatic cancer cells after transfected with somatostatin receptor type 2 gene.

Zheng-Ren Liu1, Ren-Yi Qin, Gao-Song Wu, Qing Chang, Da-Yu Wang, Sheng-Quan Zou, Fa-Zu Qiu.   

Abstract

AIM: To observe the effect of octreotide on apoptosis rate of human pancreatic cancer cells PC-3 after transfected with somatostatin receptor type 2 (SST2) gene.
METHODS: SST2 plasmid was transfected into PC-3 cells by liposome. Result of transfection was detected by immunocytochemical staining and Western blotting. Apoptosis rates of PC-3 cells under different dosages of octreotide were measured by MTT assay and flow cytometry (FCM).
RESULTS: Apoptosis rate caused by octreotide of transfected PC-3 cells was 7.56+/-1.06% at the dosage of 0.20 microg/mL, 9.25+/-1.73% at the dosage of 0.40 microg/mL and 14.18+/-2.71% at the dosage of 0.80 microg/mL. Apoptosis rate caused by octreotide of non-transfected PC-3 cells was 5.76+/-0.75% at the dosage of 0.20 microg/mL, 6.69+/-0.80% at the dosage of 0.40 microg/mL and 7.26+/-1.28% at the dosage of 0.80 microg/mL. Transfected PC-3 cells growth inhibition rate caused by octreotide was 9.36+/-1.34% at the dosage of 0.20 microg/mL, 12.03+/-1.44% at the dosage of 0.40 microg/mL and 20.23+/-4.21% at the dosage of 0.80 microg/mL. Non-transfected PC-3 cells growth inhibition rate caused by octreotide was 6.44+/-0.66% at the dosage of 0.20 microg/mL, 7.65+/-0.88% at the dosage of 0.40 microg/mL and 9.29+/-1.32% at the dosage of 0.80 microg/mL. We found that octreotide caused higher apoptosis rate and inhibition rate in transfected groups than in non-transfected groups (P<0.05) at the tested dosages (0.20, 0.40 and 0.80 microg/mL).
CONCLUSION: Deficiency of SST2 was probably the major reason why octreotide had little effect on PC-3 cells. Transfecting SST2 gene could strengthen the ability of octreotide of killing PC-3 cells. It provided an experimental evidence for using both octreotide and transfection with SST2 gene on clinical treatment of pancreatic cancer.

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Year:  2004        PMID: 15259086      PMCID: PMC4724970          DOI: 10.3748/wjg.v10.i15.2292

Source DB:  PubMed          Journal:  World J Gastroenterol        ISSN: 1007-9327            Impact factor:   5.742


  15 in total

1.  sst2 somatostatin receptor expression reverses tumorigenicity of human pancreatic cancer cells.

Authors:  N Delesque; L Buscail; J P Estève; N Saint-Laurent; C Müller; G Weckbecker; C Bruns; N Vaysse; C Susini
Journal:  Cancer Res       Date:  1997-03-01       Impact factor: 12.701

2.  Loss of sst2 somatostatin receptor gene expression in human pancreatic and colorectal cancer.

Authors:  L Buscail; N Saint-Laurent; E Chastre; J C Vaillant; C Gespach; G Capella; H Kalthoff; F Lluis; N Vaysse; C Susini
Journal:  Cancer Res       Date:  1996-04-15       Impact factor: 12.701

3.  Classification and nomenclature of somatostatin receptors.

Authors:  D Hoyer; G I Bell; M Berelowitz; J Epelbaum; W Feniuk; P P Humphrey; A M O'Carroll; Y C Patel; A Schonbrunn; J E Taylor
Journal:  Trends Pharmacol Sci       Date:  1995-03       Impact factor: 14.819

4.  Differential regulation of somatostatin receptor type 2 (sst 2) expression in AR4-2J tumor cells implanted into mice during octreotide treatment.

Authors:  S Froidevaux; E Hintermann; M Török; H R Mäcke; C Beglinger; A N Eberle
Journal:  Cancer Res       Date:  1999-08-01       Impact factor: 12.701

5.  Somatostatin receptor subtypes 2 and 4 affect seizure susceptibility and hippocampal excitatory neurotransmission in mice.

Authors:  D Moneta; C Richichi; M Aliprandi; P Dournaud; P Dutar; J M Billard; A S Carlo; C Viollet; J P Hannon; D Fehlmann; C Nunn; D Hoyer; J Epelbaum; A Vezzani
Journal:  Eur J Neurosci       Date:  2002-09       Impact factor: 3.386

6.  Regulation of stress response signaling by the N-terminal dishevelled/EGL-10/pleckstrin domain of Sst2, a regulator of G protein signaling in Saccharomyces cerevisiae.

Authors:  Scott A Burchett; Paul Flanary; Christopher Aston; Lixin Jiang; Kathleen H Young; Peter Uetz; Stanley Fields; Henrik G Dohlman
Journal:  J Biol Chem       Date:  2002-04-08       Impact factor: 5.157

Review 7.  Somatostatin receptor subtype expression in human tumors.

Authors:  L J Hofland; S W Lamberts
Journal:  Ann Oncol       Date:  2001       Impact factor: 32.976

8.  Potentiation of the anti-proliferative effects of anti-cancer drugs by octreotide in vitro and in vivo.

Authors:  G Weckbecker; F Raulf; L Tolcsvai; C Bruns
Journal:  Digestion       Date:  1996       Impact factor: 3.216

9.  Somatostatin receptor subtype 2 sensitizes human pancreatic cancer cells to death ligand-induced apoptosis.

Authors:  Julie Guillermet; Nathalie Saint-Laurent; Philippe Rochaix; Olivier Cuvillier; Thierry Levade; Andrew V Schally; Lucien Pradayrol; Louis Buscail; Christiane Susini; Corinne Bousquet
Journal:  Proc Natl Acad Sci U S A       Date:  2002-12-18       Impact factor: 11.205

10.  Treatment of advanced pancreatic cancer with the long-acting somatostatin analogue lanreotide: in vitro and in vivo results.

Authors:  M Raderer; G Hamilton; A Kurtaran; J Valencak; I Haberl; O Hoffmann; G V Kornek; F Vorbeck; M H Hejna; I Virgolini; W Scheithauer
Journal:  Br J Cancer       Date:  1999-02       Impact factor: 7.640

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