Literature DB >> 15246016

Microplate screening assay to identify inhibitors of human catechol-O-methyltransferase.

Mika Kurkela1, Antti Siiskonen, Moshe Finel, Päivi Tammela, Jyrki Taskinen, Pia Vuorela.   

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Year:  2004        PMID: 15246016     DOI: 10.1016/j.ab.2004.04.026

Source DB:  PubMed          Journal:  Anal Biochem        ISSN: 0003-2697            Impact factor:   3.365


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  8 in total

1.  Synthesis and Evaluation of Heterocyclic Catechol Mimics as Inhibitors of Catechol-O-methyltransferase (COMT).

Authors:  Scott T Harrison; Michael S Poslusney; James J Mulhearn; Zhijian Zhao; Nathan R Kett; Jeffrey W Schubert; Jeffrey Y Melamed; Timothy J Allison; Sangita B Patel; John M Sanders; Sujata Sharma; Robert F Smith; Dawn L Hall; Ronald G Robinson; Nancy A Sachs; Pete H Hutson; Scott E Wolkenberg; James C Barrow
Journal:  ACS Med Chem Lett       Date:  2015-01-26       Impact factor: 4.345

2.  Inhibition of catechol-Omicron-methyltransferase activity in human breast cancer cells enhances the biological effect of the green tea polyphenol (-)-EGCG.

Authors:  Kristin Landis-Piwowar; Di Chen; Tak Hang Chan; Q Ping Dou
Journal:  Oncol Rep       Date:  2010-08       Impact factor: 3.906

3.  Clitoria ternatea ameliorated the intracerebroventricularly injected streptozotocin induced cognitive impairment in rats: behavioral and biochemical evidence.

Authors:  Jogender Mehla; Monika Pahuja; Pooja Gupta; Shekhar Dethe; Amit Agarwal; Yogendra Kumar Gupta
Journal:  Psychopharmacology (Berl)       Date:  2013-07-06       Impact factor: 4.530

4.  SERMs attenuate estrogen-induced malignant transformation of human mammary epithelial cells by upregulating detoxification of oxidative metabolites.

Authors:  L P Madhubhani P Hemachandra; Hitisha Patel; R Esala P Chandrasena; Jaewoo Choi; Sujeewa C Piyankarage; Shuai Wang; Yijin Wang; Emily N Thayer; Robert A Scism; Bradley T Michalsen; Rui Xiong; Marton I Siklos; Judy L Bolton; Gregory R J Thatcher
Journal:  Cancer Prev Res (Phila)       Date:  2014-03-05

5.  Characterization of non-nitrocatechol pan and isoform specific catechol-O-methyltransferase inhibitors and substrates.

Authors:  Ronald G Robinson; Sean M Smith; Scott E Wolkenberg; Monika Kandebo; Lihang Yao; Christopher R Gibson; Scott T Harrison; Stacey Polsky-Fisher; James C Barrow; Peter J Manley; James J Mulhearn; Kausik K Nanda; Jeffrey W Schubert; B Wesley Trotter; Zhijian Zhao; John M Sanders; Robert F Smith; Debra McLoughlin; Sujata Sharma; Dawn L Hall; Tiffany L Walker; Jennifer L Kershner; Neetesh Bhandari; Pete H Hutson; Nancy A Sachs
Journal:  ACS Chem Neurosci       Date:  2011-11-14       Impact factor: 4.418

Review 6.  Coumarin-Based Profluorescent and Fluorescent Substrates for Determining Xenobiotic-Metabolizing Enzyme Activities In Vitro.

Authors:  Hannu Raunio; Olli Pentikäinen; Risto O Juvonen
Journal:  Int J Mol Sci       Date:  2020-07-01       Impact factor: 5.923

Review 7.  Analytical methodologies for sensing catechol-O-methyltransferase activity and their applications.

Authors:  Fang-Yuan Wang; Ping Wang; Dong-Fang Zhao; Frank J Gonzalez; Yu-Fan Fan; Yang-Liu Xia; Guang-Bo Ge; Ling Yang
Journal:  J Pharm Anal       Date:  2020-04-07

8.  A universal competitive fluorescence polarization activity assay for S-adenosylmethionine utilizing methyltransferases.

Authors:  Tiffany L Graves; Yi Zhang; John E Scott
Journal:  Anal Biochem       Date:  2007-09-29       Impact factor: 3.365

  8 in total

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