Literature DB >> 15212166

Effects of duration of ischemia and donor pretreatment with methylprednisolone or its macromolecular prodrug on the disposition of indocyanine green in cold-preserved rat livers.

Anjaneya P Chimalakonda1, Reza Mehvar.   

Abstract

PURPOSE: Cold preservation of the liver before transplantation may change uptake and excretory functions of hepatocytes. We hypothesized that an increase in the duration of preservation would result in a progressive decrease in the hepatic uptake and/or biliary excretion of indocyanine green (ICG), which would be attenuated by pharmacologic interventions.
METHODS: Donor rats (n = 40) were administered saline (control) or single 5 mg/kg doses of methylprednisolone (MP) or its liver-targeted prodrug (DMP) 2 h prior to liver harvest. Following preservation in cold University of Wisconsin solution for 0, 24, 48, or 72 h, livers were reperfused in a single-pass manner for 30 min in the presence of ICG (approximately 4 microg/ml), followed by 60 min of ICG-free perfusion. The inlet, outlet, and bile concentrations of ICG were measured periodically by high performance liquid chromatography (HPLC), and kinetic parameters were estimated.
RESULTS: Effects of duration of preservation: In unpreserved livers, a significant portion of ICG dose (16%) was effluxed from the liver during the washout period. Cold preservation for 24-72 h progressively increased (p < 0.05) the efflux of ICG (>2-fold at 72 h). Similarly, average extraction ratio showed a modest (30-40%) decrease with increasing preservation time (p < 0.05). However, biliary excretion of ICG showed the most sensitivity to the preservation time (14 to >800-fold decline). Effects of pretreatment: DMP caused significant (p < 0.05) increases in biliary ICG levels (>12-fold) and bile flow rates (6-15-fold) of preserved livers. Although MP pretreatment significantly (p < 0.05) increased (6-fold) bile flow rates in 48-h preserved livers, its effects on biliary ICG levels were not significant (p > 0.05).
CONCLUSIONS: Biliary excretion of ICG is the most sensitive kinetic parameter to prolonged cold ischemia-reperfusion injury in a rat liver perfusion model. The injury may be significantly attenuated by pharmacologic pretreatment of the liver donors.

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Year:  2004        PMID: 15212166     DOI: 10.1023/b:pham.0000029290.54167.7c

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  32 in total

Review 1.  Preservation and reperfusion injuries in liver allografts. An overview and synthesis of current studies.

Authors:  P A Clavien; P R Harvey; S M Strasberg
Journal:  Transplantation       Date:  1992-05       Impact factor: 4.939

2.  High-performance size-exclusion chromatographic analysis of dextran-methylprednisolone hemisuccinate in rat plasma.

Authors:  R Mehvar
Journal:  J Chromatogr B Biomed Sci Appl       Date:  2000-07-21

3.  Detection of graft nonfunction after liver transplantation by assessment of indocyanine green kinetics.

Authors:  C G Krenn; B Schäfer; G A Berlakovich; R Steininger; H Steltzer; C K Spiss
Journal:  Anesth Analg       Date:  1998-07       Impact factor: 5.108

4.  Multidrug resistance p-glycoprotein 2 is essential for the biliary excretion of indocyanine green.

Authors:  L Huang; M Vore
Journal:  Drug Metab Dispos       Date:  2001-05       Impact factor: 3.922

5.  Simultaneous analysis of methylprednisolone, methylprednisolone succinate, and endogenous corticosterone in rat plasma.

Authors:  R Mehvar; R O Dann; D A Hoganson
Journal:  J Pharm Biomed Anal       Date:  2000-07       Impact factor: 3.935

6.  Kupffer cell-independent acute hepatocellular oxidative stress and decreased bile formation in post-cold-ischemic rat liver.

Authors:  Y Kumamoto; M Suematsu; M Shimazu; Y Kato; T Sano; N Makino; K I Hirano; M Naito; G Wakabayashi; Y Ishimura; M Kitajima
Journal:  Hepatology       Date:  1999-12       Impact factor: 17.425

7.  Effects of LPS on transport of indocyanine green and alanine uptake in perfused rat liver.

Authors:  M Lund; L Kang; N Tygstrup; A W Wolkoff; P Ott
Journal:  Am J Physiol       Date:  1999-07

Review 8.  Role of hepatocytes and bile duct cells in preservation-reperfusion injury of liver grafts.

Authors:  M Kukan; P S Haddad
Journal:  Liver Transpl       Date:  2001-05       Impact factor: 5.799

9.  Stability of indocyanine green in human serum stored at -20 and -70 degrees C.

Authors:  C March; M H Adams; W Garnett; H T Karnes
Journal:  Ther Drug Monit       Date:  1994-12       Impact factor: 3.681

10.  Effect of H2-receptor antagonists on steady-state extraction of indocyanine green and lidocaine by the perfused rat liver.

Authors:  R K Roberts; C A Heath; R F Johnson; K V Speeg; S Schenker
Journal:  J Lab Clin Med       Date:  1986-02
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  3 in total

1.  Multidrug donor preconditioning prevents cold liver preservation and reperfusion injury.

Authors:  Mohammed Reza Moussavian; Claudia Scheuer; Michael Schmidt; Otto Kollmar; Matthias Wagner; Maximilian von Heesen; Martin K Schilling; Michael D Menger
Journal:  Langenbecks Arch Surg       Date:  2010-06-27       Impact factor: 3.445

2.  Effects of methylprednisolone and its liver-targeted dextran prodrug on ischemia-reperfusion injury in a rat liver transplantation model.

Authors:  Anjaneya P Chimalakonda; Reza Mehvar
Journal:  Pharm Res       Date:  2007-10-06       Impact factor: 4.200

3.  Trimetazidine: is it a promising drug for use in steatotic grafts?

Authors:  Ismail Ben Mosbah; Araní Casillas-Ramírez; Carme Xaus; Anna Serafín; Joan Roselló-Catafau; Carmen Peralta
Journal:  World J Gastroenterol       Date:  2006-02-14       Impact factor: 5.742

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