Literature DB >> 15173840

Antimalarial drug discovery: efficacy models for compound screening.

David A Fidock1, Philip J Rosenthal, Simon L Croft, Reto Brun, Solomon Nwaka.   

Abstract

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Year:  2004        PMID： 15173840     DOI： 10.1038/nrd1416

Source DB:  PubMed          Journal:  Nat Rev Drug Discov        ISSN： 1474-1776            Impact factor:   84.694


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  204 in total

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Authors:  Ramesh Gujjar; Farah El Mazouni; Karen L White; John White; Sharon Creason; David M Shackleford; Xiaoyi Deng; William N Charman; Ian Bathurst; Jeremy Burrows; David M Floyd; David Matthews; Frederick S Buckner; Susan A Charman; Margaret A Phillips; Pradipsinh K Rathod
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2.  Fighting malaria at the crossroads.

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Journal:  EMBO Rep       Date:  2004-09       Impact factor: 8.807

3.  Self-microemulsifiyng suppository formulation of β-artemether.

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4.  Substrate mapping and inhibitor profiling of falcipain-2, falcipain-3 and berghepain-2: implications for peptidase anti-malarial drug discovery.

Authors:  Manoj K Ramjee; Nicholas S Flinn; Tracy P Pemberton; Martin Quibell; Yikang Wang; John P Watts
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Review 5.  Antiplasmodial marine natural products in the perspective of current chemotherapy and prevention of malaria: a review.

Authors:  Dominique Laurent; Francesco Pietra
Journal:  Mar Biotechnol (NY)       Date:  2006-03-30       Impact factor: 3.619

6.  Antiplasmodial activity of Indigofera spicata root extract against Plasmodium berghei infection in mice.

Authors:  Eshetie Melese Birru; Mestayet Geta; Abyot Endale Gurmu
Journal:  Malar J       Date:  2017-05-16       Impact factor: 2.979

7.  In vivo anti-malarial effect of the beta-amino alcohol 1t on Plasmodium berghei.

Authors:  N Bahamontes-Rosa; K Bucher; J Held; A Robin; W H Hoffmann; S L Flitsch; P G Kremsner; J F J Kun
Journal:  Parasitol Res       Date:  2009-01-27       Impact factor: 2.289

8.  Analogs of natural aminoacyl-tRNA synthetase inhibitors clear malaria in vivo.

Authors:  Eva Maria Novoa; Noelia Camacho; Anna Tor; Barrie Wilkinson; Steven Moss; Patricia Marín-García; Isabel G Azcárate; José M Bautista; Adam C Mirando; Christopher S Francklyn; Sònia Varon; Miriam Royo; Alfred Cortés; Lluís Ribas de Pouplana
Journal:  Proc Natl Acad Sci U S A       Date:  2014-12-08       Impact factor: 11.205

9.  Identification and deconvolution of cross-resistance signals from antimalarial compounds using multidrug-resistant Plasmodium falciparum strains.

Authors:  Monika Chugh; Christian Scheurer; Sibylle Sax; Elizabeth Bilsland; Donelly A van Schalkwyk; Kathryn J Wicht; Natalie Hofmann; Anil Sharma; Sridevi Bashyam; Shivendra Singh; Stephen G Oliver; Timothy J Egan; Pawan Malhotra; Colin J Sutherland; Hans-Peter Beck; Sergio Wittlin; Thomas Spangenberg; Xavier C Ding
Journal:  Antimicrob Agents Chemother       Date:  2014-12-08       Impact factor: 5.191

Review 10.  Malaria: progress, perils, and prospects for eradication.

Authors:  Brian M Greenwood; David A Fidock; Dennis E Kyle; Stefan H I Kappe; Pedro L Alonso; Frank H Collins; Patrick E Duffy
Journal:  J Clin Invest       Date:  2008-04       Impact factor: 14.808
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