Literature DB >> 15125960

New highly selective inhibitors of class II fructose-1,6-bisphosphate aldolases.

Matthieu Fonvielle1, Philippe Weber, Kasia Dabkowska, Michel Therisod.   

Abstract

Phosphoglycolo amidoxime and phosphoglycolo hydrazide, two new derivatives of phosphoglycolic acid, were synthesised and successfully tested as selective competitive inhibitors of class II FBP-aldolases.

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Year:  2004        PMID： 15125960     DOI： 10.1016/j.bmcl.2004.03.040

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

1.  Rational design, synthesis, and evaluation of new selective inhibitors of microbial class II (zinc dependent) fructose bis-phosphate aldolases.

Authors:  Racha Daher; Mathieu Coinçon; Matthieu Fonvielle; Petra M Gest; Marcelo E Guerin; Mary Jackson; Jurgen Sygusch; Michel Therisod
Journal:  J Med Chem       Date:  2010-11-11       Impact factor: 7.446

Review 2.  Targeting Metalloenzymes for Therapeutic Intervention.

Authors:  Allie Y Chen; Rebecca N Adamek; Benjamin L Dick; Cy V Credille; Christine N Morrison; Seth M Cohen
Journal:  Chem Rev       Date:  2018-09-07       Impact factor: 60.622

3.  Active site loop dynamics of a class IIa fructose 1,6-bisphosphate aldolase from Mycobacterium tuberculosis.

Authors:  Scott D Pegan; Kamolchanok Rukseree; Glenn C Capodagli; Erica A Baker; Olga Krasnykh; Scott G Franzblau; Andrew D Mesecar
Journal:  Biochemistry       Date:  2013-01-18       Impact factor: 3.162

4.  A noncompetitive inhibitor for Mycobacterium tuberculosis's class IIa fructose 1,6-bisphosphate aldolase.

Authors:  Glenn C Capodagli; Wafik G Sedhom; Mary Jackson; Kateri A Ahrendt; Scott D Pegan
Journal:  Biochemistry       Date:  2013-12-24       Impact factor: 3.162

5.  Structural basis for catalysis of a tetrameric class IIa fructose 1,6-bisphosphate aldolase from Mycobacterium tuberculosis.

Authors:  Scott D Pegan; Kamolchanok Rukseree; Scott G Franzblau; Andrew D Mesecar
Journal:  J Mol Biol       Date:  2009-01-10       Impact factor: 5.469

6.  Structural and functional characterization of methicillin-resistant Staphylococcus aureus's class IIb fructose 1,6-bisphosphate aldolase.

Authors:  Glenn C Capodagli; Stephen A Lee; Kyle J Boehm; Kristin M Brady; Scott D Pegan
Journal:  Biochemistry       Date:  2014-11-21       Impact factor: 3.162
  6 in total

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