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55 in total

1. Synthesis and structure-activity relationship studies of 4-((2-hydroxy-3-methoxybenzyl)amino)benzenesulfonamide derivatives as potent and selective inhibitors of 12-lipoxygenase.

Authors: Diane K Luci; J Brian Jameson; Adam Yasgar; Giovanni Diaz; Netra Joshi; Auric Kantz; Kate Markham; Steve Perry; Norine Kuhn; Jennifer Yeung; Edward H Kerns; Lena Schultz; Michael Holinstat; Jerry L Nadler; David A Taylor-Fishwick; Ajit Jadhav; Anton Simeonov; Theodore R Holman; David J Maloney
Journal: J Med Chem Date: 2014-01-06 Impact factor: 7.446

Review 2. Prodrug approaches for CNS delivery.

Authors: Jarkko Rautio; Krista Laine; Mikko Gynther; Jouko Savolainen
Journal: AAPS J Date: 2008-02-05 Impact factor: 4.009

3. Preclinical development of drug delivery systems for paclitaxel-based cancer chemotherapy.

Authors: Feihu Wang; Michael Porter; Alexandros Konstantopoulos; Pengcheng Zhang; Honggang Cui
Journal: J Control Release Date: 2017-09-25 Impact factor: 9.776

4. Human carboxymethylenebutenolidase as a bioactivating hydrolase of olmesartan medoxomil in liver and intestine.

Authors: Tomoko Ishizuka; Izumi Fujimori; Mitsunori Kato; Chisa Noji-Sakikawa; Motoko Saito; Yasushi Yoshigae; Kazuishi Kubota; Atsushi Kurihara; Takashi Izumi; Toshihiko Ikeda; Osamu Okazaki
Journal: J Biol Chem Date: 2010-02-19 Impact factor: 5.157

Review 5. Predicting drug metabolism: experiment and/or computation?

Authors: Johannes Kirchmair; Andreas H Göller; Dieter Lang; Jens Kunze; Bernard Testa; Ian D Wilson; Robert C Glen; Gisbert Schneider
Journal: Nat Rev Drug Discov Date: 2015-04-24 Impact factor: 84.694

6. Homology modeling and metabolism prediction of human carboxylesterase-2 using docking analyses by GriDock: a parallelized tool based on AutoDock 4.0.

Authors: Giulio Vistoli; Alessandro Pedretti; Angelica Mazzolari; Bernard Testa
Journal: J Comput Aided Mol Des Date: 2010-07-11 Impact factor: 3.686

7. Population pharmacokinetics of modafinil acid and estimation of the metabolic conversion of modafinil into modafinil acid in 5 major ethnic groups of China.

Authors: Ke-hua Wu; Tao Guo; Chen-hui Deng; Zheng Guan; Liang Li; Tian-yan Zhou; Wei Lu
Journal: Acta Pharmacol Sin Date: 2012-10-29 Impact factor: 6.150

8. Degradation of poly(β-amino ester) gels in alcohols through transesterification: A method to conjugate drugs to polymer matrices.

Authors: Prachi Gupta; Caroline Lacerda; Vinod Patil; Dipti Biswal; Paritosh Wattamwar; J Zach Hilt; Thomas D Dziubla
Journal: J Polym Sci A Polym Chem Date: 2017-03-25 Impact factor: 2.702

9. Alkyne Ligation Handles: Propargylation of Hydroxyl, Sulfhydryl, Amino, and Carboxyl Groups via the Nicholas Reaction.

Authors: Sarah M Wells; John C Widen; Daniel A Harki; Kay M Brummond
Journal: Org Lett Date: 2016-08-29 Impact factor: 6.005

10. Enhancing the intestinal absorption of molecules containing the polar guanidino functionality: a double-targeted prodrug approach.

Authors: Jing Sun; Arik Dahan; Gordon L Amidon
Journal: J Med Chem Date: 2010-01-28 Impact factor: 7.446