Literature DB >> 15040739

Full orthogonality between Dde and Fmoc: the direct synthesis of PNA--peptide conjugates.

Juan Jose Díaz-Mochón1, Laurent Bialy, Mark Bradley.   

Abstract

New deprotection conditions for the Dde amine protecting group that are fully orthogonal to Fmoc are described and successfully applied to the dual synthesis of PNA-peptide conjugates.

Entities:  

Year:  2004        PMID： 15040739     DOI： 10.1021/ol049905y

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  19 in total

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4.  Histone-Mimetic Gold Nanoparticles as Versatile Scaffolds for Gene Transfer and Chromatin Analysis.

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Journal:  Bioconjug Chem       Date:  2018-10-29       Impact factor: 4.774

5.  One-Bead-Two-Compound Thioether Bridged Macrocyclic γ-AApeptide Screening Library against EphA2.

Authors:  Yan Shi; Sridevi Challa; Peng Sang; Fengyu She; Chunpu Li; Geoffrey M Gray; Alekhya Nimmagadda; Peng Teng; Timothy Odom; Yan Wang; Arjan van der Vaart; Qi Li; Jianfeng Cai
Journal:  J Med Chem       Date:  2017-11-14       Impact factor: 7.446

6.  A family of bioreducible poly(disulfide amine)s for gene delivery.

Authors:  Mei Ou; Rongzuo Xu; Sun Hwa Kim; David A Bull; Sung Wan Kim
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Authors:  Konstantin Andreev; Christopher Bianchi; Jonas S Laursen; Linda Citterio; Line Hein-Kristensen; Lone Gram; Ivan Kuzmenko; Christian A Olsen; David Gidalevitz
Journal:  Biochim Biophys Acta       Date:  2014-05-28

8.  Synthesis of peptide nucleic acid FRET probes via an orthogonally protected building block for post-synthetic labeling of peptide nucleic acids at the 5-position of uracil.

Authors:  Bereket Y Oquare; John-Stephen Taylor
Journal:  Bioconjug Chem       Date:  2008-11-19       Impact factor: 4.774

9.  Melanoma targeting with alpha-melanocyte stimulating hormone analogs labeled with fac-[99mTc(CO)3]+: effect of cyclization on tumor-seeking properties.

Authors:  Paula D Raposinho; Catarina Xavier; João D G Correia; Soraia Falcão; Paula Gomes; Isabel Santos
Journal:  J Biol Inorg Chem       Date:  2008-01-08       Impact factor: 3.358

10.  Synthetic Antibody Mimics Based on Cancer-Targeting Immunostimulatory Peptides.

Authors:  Dante Descalzi-Montoya; Rachel A Montel; Keith Smith; Eugenia Dziopa; Andrieh Darwich; Zheng Yang; Constantine Bitsaktsis; Robert Korngold; David Sabatino
Journal:  Chembiochem       Date:  2020-11-02       Impact factor: 3.164
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