Literature DB >> 14748820

Sildenafil does not improve nitric oxide-mediated endothelium-dependent vascular responses in smokers.

Victor Dishy1, Paul A Harris, Rosanna Pierce, Harish C Prasad, Gbenga Sofowora, Holly L Bonar, Alastair J J Wood, C Michael Stein.   

Abstract

AIMS: To examine the hypothesis that sildenafil, a phosphodiesterase type 5 inhibitor that inhibits cGMP breakdown, could enhance nitric oxide-mediated vasodilation and reverse endothelial dysfunction in chronic smokers.
METHODS: Flow-mediated dilation of the brachial artery and forearm postischemic reactive hyperemia (both nitric oxide-mediated responses) were measured before and after sildenafil 50 mg and placebo in a double-blind, randomized, crossover study in 9 men who were chronic smokers (21 +/- 3 pack years).
RESULTS: There was no significant change in flow-mediated dilation after either sildenafil (0.18%, 95%CI -1.7-2%) or placebo (0.24%, 95%CI -2.8-3.3%) (P = 0.88 and 0.8, respectively). Sildenafil had no significant effect on resting forearm blood flow or postischemic reactive hyperemia (P = 0.39 and 0.7, respectively). Resting heart rate and blood pressure were unaffected by sildenafil.
CONCLUSIONS: Acute sildenafil administration did not improve endothelial function in chronic smoking men.

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Year:  2004        PMID: 14748820      PMCID: PMC1884430          DOI: 10.1046/j.1365-2125.2003.01974.x

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN: 0306-5251            Impact factor:   4.335


  16 in total

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