| Literature DB >> 14741297 |
Alexander Alanine1, Lilli Anselm, Lucinda Steward, Stefan Thomi, Walter Vifian, Michael D Groaning.
Abstract
The synthesis and in vitro structure-activity relationships (SAR) of a series of triazoles as A(2A) receptor antagonists is reported. This resulted in the identification of potent, selective and permeable 1,2,4-triazoles such as 42 for further optimization and evaluation in vivo.Entities:
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Year: 2004 PMID： 14741297 DOI： 10.1016/j.bmcl.2003.09.095
Source DB: PubMed Journal: Bioorg Med Chem Lett ISSN： 0960-894X Impact factor: 2.823