Literature DB >> 14737353

Facile palladium-catalysed synthesis of 1-aryl-1H-indazoles from 2-bromobenzaldehydes and arylhydrazines.

Chan Sik Cho1, Dong Kwon Lim, Nam Ho Heo, Tae-Jeong Kim, Sang Chul Shim.   

Abstract

2-Bromobenzaldehydes react with arylhydrazines in toluene at 100 [degree]C in the presence of a catalytic amount of a palladium catalyst and phosphorus chelating ligands such as 1,1[prime or minute]-bis(diphenylphosphino)ferrocene and 1,3-bis(diphenylphosphino)propane along with NaO-t-Bu to afford 1-aryl-1H-indazoles in good yields.

Entities:  

Year:  2003        PMID: 14737353     DOI: 10.1039/b312154m

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN: 1359-7345            Impact factor:   6.222


  2 in total

1.  Synthesis of 1H-Indazoles via Silver(I)-Mediated Intramolecular Oxidative C-H Bond Amination.

Authors:  Areum Park; Kyu-Sung Jeong; Hyuk Lee; Hyunwoo Kim
Journal:  ACS Omega       Date:  2021-02-23

2.  Synthesis of N-phenyl- and N-thiazolyl-1H-indazoles by copper-catalyzed intramolecular N-arylation of ortho-chlorinated arylhydrazones.

Authors:  Yara Cristina Marchioro Barbosa; Guilherme Caneppele Paveglio; Claudio Martin Pereira de Pereira; Sidnei Moura; Cristiane Storck Schwalm; Gleison Antonio Casagrande; Lucas Pizzuti
Journal:  Beilstein J Org Chem       Date:  2022-08-23       Impact factor: 2.544

  2 in total

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