Literature DB >> 14725444

Facile preparation of beta-fluoro amines by the reaction of aziridines with potassium fluoride dihydrate in the presence of Bu4NHSO4.

Ren-Hua Fan1, Yong-Gui Zhou, Wan-Xuan Zhang, Xue-Long Hou, Li-Xin Dai.   

Abstract

Potassium fluoride combined with tetrabutylammonium bisulfate is an efficient reagent to convert a variety of aziridines derived from cyclic and acyclic alkenes to beta-fluoro amine derivatives in high yield.

Entities:  

Year:  2004        PMID： 14725444     DOI： 10.1021/jo034895k

Source DB:  PubMed          Journal:  J Org Chem        ISSN： 0022-3263            Impact factor:   4.354


  6 in total

1.  Multifaceted Ion Exchange Resin-Supported Hydrogen Fluoride: A Path to Flow Hydrofluorination.

Authors:  Zhichao Lu; Bhvandip S Bajwa; Otome E Okoromoba; Gerald B Hammond; Bo Xu
Journal:  Green Chem       Date:  2018-12-26       Impact factor: 10.182

2.  Highly efficient diastereoselective reduction of alpha-fluoroimines.

Authors:  Roy M Malamakal; Whitney R Hess; Todd A Davis
Journal:  Org Lett       Date:  2010-05-21       Impact factor: 6.005

3.  Achieving regio- and stereo-control in the fluorination of aziridines under acidic conditions.

Authors:  Otome E Okoromoba; Zhou Li; Nicole Robertson; Mark S Mashuta; Uenifer R Couto; Cláudio F Tormena; Bo Xu; Gerald B Hammond
Journal:  Chem Commun (Camb)       Date:  2016-11-08       Impact factor: 6.222

4.  Efficient regioselective ring opening of activated aziridine-2-carboxylates with [(18)f]fluoride.

Authors:  Christina Schjoeth-Eskesen; Paul Robert Hansen; Andreas Kjaer; Nic Gillings
Journal:  ChemistryOpen       Date:  2014-11-21       Impact factor: 2.911

Review 5.  Organocatalyzed enantioselective desymmetrization of aziridines and epoxides.

Authors:  Ping-An Wang
Journal:  Beilstein J Org Chem       Date:  2013-08-15       Impact factor: 2.883

6.  Multigramme synthesis and asymmetric dihydroxylation of a 4-fluorobut-2E-enoate.

Authors:  James A B Laurenson; John A Parkinson; Jonathan M Percy; Giuseppe Rinaudo; Ricard Roig
Journal:  Beilstein J Org Chem       Date:  2013-11-26       Impact factor: 2.883
  6 in total

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