Literature DB >> 14634678

Effects of a lipase inhibitor (Orlistat) on cholecystokinin and appetite in response to a high-fat meal.

J H Goedecke1, M Barsdorf, C Beglinger, N S Levitt, E V Lambert.   

Abstract

OBJECTIVE: To examine the short-term effects of a lipase inhibitor (Orlistat) on physiological and behavioural measures of appetite in response to a high-fat meal.
DESIGN: Randomised, single blind, placebo-controlled, crossover trial.
SUBJECTS: A total of 19 healthy nonobese male subjects. PROCEDURES: After an overnight fast, subjects ingested a test meal of 2940 kJ (60% fat, 30% CHO, 10% protein) with Orlistat (120 mg) or a placebo, separated by 2 weeks. Appetite, as assessed by a standard line scale, and plasma cholecystokinin (CCK) concentrations were measured prior to and every hour after the test meal for 4 h. Thereafter, subjects ingested a quantified, but self-selected portion of a standardised lunch (15% protein, 37% fat and 45% CHO), before completing a final line scale questionnaire.
RESULTS: The CCK response to the test meal was negatively correlated with BMI in both the Orlistat and placebo trials (R=-0.69 and -0.65, P<0.01). Orlistat administration did not significantly alter the CCK response to the test meal (6.30+/-3.27 vs 7.36+/-3.94 pM min, for Orlistat and placebo, P=0.193). Similarly, the line scale measures of appetite and subsequent intake (520+/-205 vs 554+/-197 g, P=0.48) were not different between the trials.
CONCLUSION: Orlistat administration did not alter short-term physiological or behavioural measures of satiety in response to a high-fat meal in healthy, nonobese subjects. The CCK response to a test meal may be partly determined by BMI.

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Year:  2003        PMID: 14634678     DOI: 10.1038/sj.ijo.0802436

Source DB:  PubMed          Journal:  Int J Obes Relat Metab Disord


  6 in total

Review 1.  Orlistat-associated adverse effects and drug interactions: a critical review.

Authors:  Theodosios D Filippatos; Christos S Derdemezis; Irene F Gazi; Eleni S Nakou; Dimitri P Mikhailidis; Moses S Elisaf
Journal:  Drug Saf       Date:  2008       Impact factor: 5.606

Review 2.  Benefit-risk assessment of orlistat in the treatment of obesity.

Authors:  Priya Sumithran; Joseph Proietto
Journal:  Drug Saf       Date:  2014-08       Impact factor: 5.606

3.  Chloroplast membranes retard fat digestion and induce satiety: effect of biological membranes on pancreatic lipase/co-lipase.

Authors:  Per-Ake Albertsson; Rickard Köhnke; Sinan C Emek; Jie Mei; Jens F Rehfeld; Hans-Erik Akerlund; Charlotte Erlanson-Albertsson
Journal:  Biochem J       Date:  2007-02-01       Impact factor: 3.857

4.  Fasting and meal-induced CCK and PP secretion following intragastric balloon treatment for obesity.

Authors:  Elisabeth M H Mathus-Vliegen; Gerrit H de Groot
Journal:  Obes Surg       Date:  2013-05       Impact factor: 4.129

Review 5.  Gut fat signaling and appetite control with special emphasis on the effect of thylakoids from spinach on eating behavior.

Authors:  C J Rebello; C E O'Neil; F L Greenway
Journal:  Int J Obes (Lond)       Date:  2015-07-31       Impact factor: 5.095

6.  The Use of Green Leaf Membranes to Promote Appetite Control, Suppress Hedonic Hunger and Loose Body Weight.

Authors:  Charlotte Erlanson-Albertsson; Per-Åke Albertsson
Journal:  Plant Foods Hum Nutr       Date:  2015-09       Impact factor: 3.921

  6 in total

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