Literature DB >> 1442957

Delayed endometrial maturation induced by daily administration of the antiprogestin RU 486: a potential new contraceptive strategy.

M C Batista1, T P Cartledge, A W Zellmer, M J Merino, C Axiotis, D L Loriaux, L K Nieman.   

Abstract

OBJECTIVE: Our objective was to determine if a progesterone antagonist might interdict the development of a secretory endometrium. STUDY
DESIGN: Eleven normally cycling women not at risk for pregnancy received RU 486 (1 mg/day orally) or placebo throughout one menstrual cycle in a randomized, double-blind, crossover fashion. Estradiol, progesterone, and placental protein 14 were measured every 3 days; luteinizing hormone was measured until the midcycle surge was detected. An endometrial biopsy was performed on luteal phase day 7 to 9 and interpreted with Noyes' criteria. Differences between treatment groups were analyzed by the Student t test.
RESULTS: RU 486 delayed ovulation, retarded endometrial maturation, and reduced peak levels of placental protein 14 without affecting gonadal steroid production. The abnormalities in endometrial morphology and function are similar to those seen in infertile women with luteal phase defects.
CONCLUSION: We hypothesize that this regimen of antiprogestin administration may prevent implantation and offer a novel strategy for fertility control.

Entities:  

Keywords:  Biology; Clinical Research; Economic Factors; Endocrine System; Endometrial Effects; Endometrium; Genitalia; Genitalia, Female; Hormone Antagonists; Hormones; Menstrual Cycle; Menstruation; Physiology; Reproduction; Research And Development; Research Methodology; Ru-486--administraction and dosage; Ru-486--pharmacodynamics; Ru-486--therapeutic use; Technology; Urogenital System; Uterus

Mesh:

Substances:

Year:  1992        PMID: 1442957     DOI: 10.1016/s0002-9378(11)91627-5

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  4 in total

1.  Clinical pharmacokinetics of mifepristone.

Authors:  O Heikinheimo
Journal:  Clin Pharmacokinet       Date:  1997-07       Impact factor: 6.447

2.  Efficacy and tolerability of CDB-2914 treatment for symptomatic uterine fibroids: a randomized, double-blind, placebo-controlled, phase IIb study.

Authors:  Lynnette K Nieman; Wendy Blocker; Tonja Nansel; Sheila Mahoney; James Reynolds; Diana Blithe; Robert Wesley; Alicia Armstrong
Journal:  Fertil Steril       Date:  2010-11-05       Impact factor: 7.329

3.  PXR mediates mifepristone-induced hepatomegaly in mice.

Authors:  Xin-Peng Yao; Ting-Ying Jiao; Yi-Ming Jiang; Shi-Cheng Fan; Ying-Yuan Zhao; Xiao Yang; Yue Gao; Fei Li; Yan-Ying Zhou; Pan-Pan Chen; Min Huang; Hui-Chang Bi
Journal:  Acta Pharmacol Sin       Date:  2021-03-29       Impact factor: 6.150

4.  Elevated serum progesterone/ MII oocyte ratio on the day of human chorionic gonadotropin administration can predict impaired endometrial receptivity.

Authors:  Abbas Aflatoonian; Robab Davar; Farzaneh Hojjat
Journal:  Iran J Reprod Med       Date:  2014-06
  4 in total

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