Literature DB >> 14406754

Compounds related to pethidine-IV. New general chemical methods of increasing the analgesic activity of pethidine.

P A JANSSEN, N B EDDY.   

Abstract

Entities:  

Keywords:  MEPERIDINE/anesthesia and analgesia

Mesh：

Substances：

Year:  1960        PMID： 14406754     DOI： 10.1021/jm50008a003

Source DB:  PubMed          Journal:  J Med Pharm Chem        ISSN： 0095-9065


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  6 in total

1.  Opioids and efflux transporters. Part 1: P-glycoprotein substrate activity of N-substituted analogs of meperidine.

Authors:  Susan L Mercer; Hazem E Hassan; Christopher W Cunningham; Natalie D Eddington; Andrew Coop
Journal:  Bioorg Med Chem Lett       Date:  2006-12-21       Impact factor: 2.823

2.  Opioid activity and distribution of fentanyl metabolites.

Authors:  E Schneider; K Brune
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1986-11       Impact factor: 3.000

3.  Opioids and efflux transporters. Part 3: P-glycoprotein substrate activity of 3-hydroxyl addition to meperidine analogs.

Authors:  Susan L Mercer; Christopher W Cunningham; Natalie D Eddington; Andrew Coop
Journal:  Bioorg Med Chem Lett       Date:  2008-04-25       Impact factor: 2.823

4.  Evaluation of the P-glycoprotein (Abcb1) affinity status of a series of morphine analogs: comparative study with meperidine analogs to identify opioids with minimal P-glycoprotein interactions.

Authors:  Hazem E Hassan; Susan L Mercer; Christopher W Cunningham; Andrew Coop; Natalie D Eddington
Journal:  Int J Pharm       Date:  2009-04-05       Impact factor: 5.875

5.  An efficient, optimized synthesis of fentanyl and related analogs.

Authors:  Carlos A Valdez; Roald N Leif; Brian P Mayer
Journal:  PLoS One       Date:  2014-09-18       Impact factor: 3.240

6.  Structural modification of fentanyls for their retrospective identification by gas chromatographic analysis using chloroformate chemistry.

Authors:  Carlos A Valdez; Roald N Leif; Robert D Sanner; Todd H Corzett; Mark L Dreyer; Katelyn E Mason
Journal:  Sci Rep       Date:  2021-11-18       Impact factor: 4.996
  6 in total

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