Literature DB >> 13491589

Inhibition of lactic acid dehydrogenase by fluoropyruvic acid.

H BUSCH, P V NAIR.   

Abstract

Entities:  

Keywords:  DEHYDROGENASES/antagonists; PYRUVATES/effects

Mesh:

Substances:

Year:  1957        PMID: 13491589

Source DB:  PubMed          Journal:  J Biol Chem        ISSN: 0021-9258            Impact factor:   5.157


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  4 in total

1.  Semipermeable membranes for improving the histochemical demonstration of enzyme activities in tissue sections. 3. Lactate dehydrogenase.

Authors:  A E Meijer
Journal:  Histochemie       Date:  1973-05-22

2.  Metabolic plasticity underpins innate and acquired resistance to LDHA inhibition.

Authors:  Aaron Boudreau; Hans E Purkey; Anna Hitz; Kirk Robarge; David Peterson; Sharada Labadie; Mandy Kwong; Rebecca Hong; Min Gao; Christopher Del Nagro; Raju Pusapati; Shuguang Ma; Laurent Salphati; Jodie Pang; Aihe Zhou; Tommy Lai; Yingjie Li; Zhongguo Chen; Binqing Wei; Ivana Yen; Steve Sideris; Mark McCleland; Ron Firestein; Laura Corson; Alex Vanderbilt; Simon Williams; Anneleen Daemen; Marcia Belvin; Charles Eigenbrot; Peter K Jackson; Shiva Malek; Georgia Hatzivassiliou; Deepak Sampath; Marie Evangelista; Thomas O'Brien
Journal:  Nat Chem Biol       Date:  2016-08-01       Impact factor: 15.040

3.  Discovery of human lactate dehydrogenase A (LDHA) inhibitors as anticancer agents to inhibit the proliferation of MG-63 osteosarcoma cells.

Authors:  Aiping Fang; Qi Zhang; Haibo Fan; Yaying Zhou; Yuqin Yao; Yue Zhang; Xiaojun Huang
Journal:  Medchemcomm       Date:  2017-07-07       Impact factor: 3.597

4.  Development of a novel lactate dehydrogenase A inhibitor with potent antitumor activity and immune activation.

Authors:  Mengyan Du; Ting Yu; Qinjinge Zhan; Han Li; Yiping Zou; Meiyu Geng; Tao Meng; Zuoquan Xie
Journal:  Cancer Sci       Date:  2022-07-11       Impact factor: 6.518

  4 in total

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