Literature DB >> 1323683

5'-Azido-delta 8-THC: a novel photoaffinity label for the cannabinoid receptor.

A Charalambous1, G Yan, D B Houston, A C Howlett, D R Compton, B R Martin, A Makriyannis.   

Abstract

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Year:  1992        PMID： 1323683     DOI： 10.1021/jm00094a023

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  8 in total

1.  2012 Division of medicinal chemistry award address. Trekking the cannabinoid road: a personal perspective.

Authors:  Alexandros Makriyannis
Journal:  J Med Chem       Date:  2014-05-01       Impact factor: 7.446

2.  Design and synthesis of the CB1 selective cannabinoid antagonist AM281: a potential human SPECT ligand.

Authors:  R Lan; J Gatley; Q Lu; P Fan; S R Fernando; N D Volkow; R Pertwee; A Makriyannis
Journal:  AAPS PharmSci       Date:  1999

3.  The role of halogen substitution in classical cannabinoids: a CB1 pharmacophore model.

Authors:  Spyros P Nikas; Jolanta Grzybowska; Demetris P Papahatjis; Avgui Charalambous; Ali R Banijamali; Ravi Chari; Pusheng Fan; Therapia Kourouli; Sonyuan Lin; Albert J Nitowski; Gilbert Marciniak; Yan Guo; Xiuyan Li; Chia-Lin J Wang; Alexandros Makriyannis
Journal:  AAPS J       Date:  2004-10-19       Impact factor: 4.009

4.  Design and synthesis of novel prostaglandin E2 ethanolamide and glycerol ester probes for the putative prostamide receptor(s).

Authors:  Erin L Shelnut; Spyros P Nikas; David F Finnegan; Nan Chiang; Charles N Serhan; Alexandros Makriyannis
Journal:  Tetrahedron Lett       Date:  2015-03-11       Impact factor: 2.415

5.  3'-functionalized adamantyl cannabinoid receptor probes.

Authors:  Go Ogawa; Marcus A Tius; Han Zhou; Spyros P Nikas; Aneetha Halikhedkar; Srikrishnan Mallipeddi; Alexandros Makriyannis
Journal:  J Med Chem       Date:  2015-03-20       Impact factor: 7.446

6.  Ligand-binding architecture of human CB2 cannabinoid receptor: evidence for receptor subtype-specific binding motif and modeling GPCR activation.

Authors:  Ying Pei; Richard W Mercier; Jenine K Anday; Ganesh A Thakur; Alexander M Zvonok; Dow Hurst; Patricia H Reggio; David R Janero; Alexandros Makriyannis
Journal:  Chem Biol       Date:  2008-11-24

7.  Synthesis and biological evaluation of indole-2-carboxamides bearing photoactivatable functionalities as novel allosteric modulators for the cannabinoid CB1 receptor.

Authors:  Chang-Jiang Qiao; Hamed I Ali; Kwang H Ahn; Srikanth Kolluru; Debra A Kendall; Dai Lu
Journal:  Eur J Med Chem       Date:  2016-05-24       Impact factor: 6.514

Review 8.  Functionalized Cannabinoid Subtype 2 Receptor Ligands: Fluorescent, PET, Photochromic and Covalent Molecular Probes.

Authors:  Filippo Basagni; Michela Rosini; Michael Decker
Journal:  ChemMedChem       Date:  2020-06-24       Impact factor: 3.466
  8 in total

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