Literature DB >> 1317926

Cyclic pentapeptide endothelin antagonists with high ETA selectivity. Potency- and solubility-enhancing modifications.

K Ishikawa, T Fukami, T Nagase, K Fujita, T Hayama, K Niiyama, T Mase, M Ihara, M Yano.   

Abstract

Entities:  

Mesh：

Substances：

Year:  1992        PMID： 1317926     DOI： 10.1021/jm00089a028

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


× No keyword cloud information.
  11 in total

1.  Clinical trials of endothelin antagonists in heart failure: publication is good for the public health.

Authors:  N F Kelland; D J Webb
Journal:  Heart       Date:  2007-01       Impact factor: 5.994

2.  Local injection of endothelin-1 produces pain-like behavior and excitation of nociceptors in rats.

Authors:  A P Gokin; M U Fareed; H L Pan; G Hans; G R Strichartz; G Davar
Journal:  J Neurosci       Date:  2001-07-15       Impact factor: 6.167

Review 3.  Role of the endothelin axis and its antagonists in the treatment of cancer.

Authors:  A Bagnato; M Loizidou; B R Pflug; J Curwen; J Growcott
Journal:  Br J Pharmacol       Date:  2011-05       Impact factor: 8.739

4.  Dual Roles for Endothelin-B Receptors in Modulating Adjuvant-Induced Inflammatory Hyperalgesia in Rats.

Authors:  Alla Khodorova; Shiping Zou; Ke Ren; Ronald Dubner; Gudarz Davar; Gary Strichartz
Journal:  Open Pain J       Date:  2009

5.  Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788.

Authors:  K Ishikawa; M Ihara; K Noguchi; T Mase; N Mino; T Saeki; T Fukuroda; T Fukami; S Ozaki; T Nagase
Journal:  Proc Natl Acad Sci U S A       Date:  1994-05-24       Impact factor: 11.205

6.  Endothelin-3 at low concentrations attenuates inflammatory responses via the endothelin B2 receptor.

Authors:  Akira Sato; Keiichi Ebina
Journal:  Inflamm Res       Date:  2013-01-31       Impact factor: 4.575

7.  Synthesis of cyclic penta- and hexapeptides: a general synthetic strategy on DAS resin.

Authors:  V Sowemimo; D Scanlon; P Jones; D J Craik
Journal:  J Protein Chem       Date:  1994-04

8.  Targeting endothelin receptors A and B attenuates the inflammatory response and improves locomotor function following spinal cord injury in mice.

Authors:  Jian Guo; Yiqiao Li; Zhennian He; Bin Zhang; Yonghuan Li; Jianghua Hu; Mingyuan Han; Yuanlin Xu; Yongfu Li; Jie Gu; Bo Dai; Zhong Chen
Journal:  Int J Mol Med       Date:  2014-04-22       Impact factor: 4.101

9.  Local injection of a selective endothelin-B receptor agonist inhibits endothelin-1-induced pain-like behavior and excitation of nociceptors in a naloxone-sensitive manner.

Authors:  Alla Khodorova; Moin U Fareed; Alexander Gokin; Gary R Strichartz; Gudarz Davar
Journal:  J Neurosci       Date:  2002-09-01       Impact factor: 6.167

10.  Discovery of Dual ETA/ETB Receptor Antagonists from Traditional Chinese Herbs through in Silico and in Vitro Screening.

Authors:  Xing Wang; Yuxin Zhang; Qing Liu; Zhixin Ai; Yanling Zhang; Yuhong Xiang; Yanjiang Qiao
Journal:  Int J Mol Sci       Date:  2016-03-16       Impact factor: 5.923
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.