Literature DB >> 12898013

Pulmonary vasodilation in the rat by insulin in vitro could indicate potential hazard for inhaled insulin.

M Aye1, W Sheedy, R Harrison, J S Thompson, A H Morice, E A Masson.   

Abstract

AIMS/HYPOTHESIS: Hypoxic pulmonary vasoconstriction is an essential mechanism to prevent hypoxaemia in lung diseases. Insulin is known to be a systemic vasodilator but its effect on the pulmonary circulation is not known. Inhaled particulate insulin can generate locally high concentrations in the lung which could be physiologically important.
METHODS: We therefore studied the effects of insulin in vitro on isolated rat pulmonary artery in a small vessel myograph.
RESULTS: We have shown that pulmonary artery vasodilatation with insulin occurs in a dose-dependent manner. Pre-constriction with PGF2alpha can be abolished (105.7+/-2.9%, mean+/-SEM) and pre-constriction with hypoxia reduced (68.9+/-6.5%) by pharmacologically relevant concentrations of insulin. The characteristic phasic vasoconstriction by pulmonary vessel to hypoxia is substantially modified, resulting in sustained vasodilatation. CONCLUSIONS/
INTERPRETATION: These effects could be clinically important for patients using inhaled insulins who have acute or occult chronic lung disease.

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Year:  2003        PMID: 12898013     DOI: 10.1007/s00125-003-1172-y

Source DB:  PubMed          Journal:  Diabetologia        ISSN: 0012-186X            Impact factor:   10.122


  7 in total

1.  Inhibition of hypoxic pulmonary vasoconstriction in isolated rat resistance arteries by atrial natriuretic peptide.

Authors:  T K Rogers; J S Thompson; A H Morice
Journal:  Eur Respir J       Date:  1997-09       Impact factor: 16.671

2.  Insulin across respiratory mucosae by aerosol delivery.

Authors:  F W Wigley; J H Londono; S H Wood; J C Shipp; R H Waldman
Journal:  Diabetes       Date:  1971-08       Impact factor: 9.461

3.  Time to peak insulin level, relative bioavailability, and effect of site of deposition of nebulized insulin in patients with noninsulin-dependent diabetes mellitus.

Authors:  B L Laube; G W Benedict; A S Dobs
Journal:  J Aerosol Med       Date:  1998

4.  Efficacy of inhaled human insulin in type 1 diabetes mellitus: a randomised proof-of-concept study.

Authors:  J S Skyler; W T Cefalu; I A Kourides; W H Landschulz; C C Balagtas; S L Cheng; R A Gelfand
Journal:  Lancet       Date:  2001-02-03       Impact factor: 79.321

5.  In vitro hypoxia on rat pulmonary artery: effects on contractions to spasmogens and role of KATP channels.

Authors:  J C Wanstall; E O'Brien
Journal:  Eur J Pharmacol       Date:  1996-05-06       Impact factor: 4.432

6.  Technosphere/Insulin--proof of concept study with a new insulin formulation for pulmonary delivery.

Authors:  S Steiner; A Pfützner; B R Wilson; O Harzer; L Heinemann; K Rave
Journal:  Exp Clin Endocrinol Diabetes       Date:  2002-01       Impact factor: 2.949

7.  Worsening of pulmonary gas exchange with nitric oxide inhalation in chronic obstructive pulmonary disease.

Authors:  J A Barberà; N Roger; J Roca; I Rovira; T W Higenbottam; R Rodriguez-Roisin
Journal:  Lancet       Date:  1996-02-17       Impact factor: 79.321

  7 in total

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