Literature DB >> 12895464

Mechanistic considerations in high-throughput screening.

Robert A Copeland1.   

Abstract

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Year:  2003        PMID： 12895464     DOI： 10.1016/s0003-2697(03)00346-4

Source DB:  PubMed          Journal:  Anal Biochem        ISSN： 0003-2697            Impact factor:   3.365


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  27 in total

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2.  Identification of two HIV inhibitors that also inhibit human RNaseH2.

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3.  Transient binding patches: a plausible concept for drug binding.

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4.  A high-throughput screen of the GTPase activity of Escherichia coli EngA to find an inhibitor of bacterial ribosome biogenesis.

Authors:  Amrita Bharat; Jan E Blanchard; Eric D Brown
Journal:  J Biomol Screen       Date:  2013-04-19

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7.  Development of a High-Throughput Screening Assay to Identify Inhibitors of the Lipid Kinase PIP5K1C.

Authors:  Brittany D Wright; Catherine Simpson; Michael Stashko; Dmitri Kireev; Emily A Hull-Ryde; Mark J Zylka; William P Janzen
Journal:  J Biomol Screen       Date:  2014-12-22

8.  Log-scale dose response of inhibitors on a chip.

Authors:  Jae Young Yun; Sachin Jambovane; Se-Kwon Kim; Sung-Hak Cho; Evert C Duin; Jong Wook Hong
Journal:  Anal Chem       Date:  2011-07-19       Impact factor: 6.986

9.  Discovery and Characterization of Two Classes of Selective Inhibitors of the Suppressor of the TCR Signaling Family of Proteins.

Authors:  Weijie Zhou; Yue Yin; Emery Smith; Jacqueline Chou; Justin Shumate; Louis Scampavia; Timothy P Spicer; Nicholas Carpino; Jarrod B French
Journal:  ACS Infect Dis       Date:  2018-12-14       Impact factor: 5.084

10.  Screening of small molecule interactor library by using in-cell NMR spectroscopy (SMILI-NMR).

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