Literature DB >> 12856409

A quantitative model of ligand binding to the glutamate site of the GluR2 subunit of AMPA receptor.

I G Tikhonova1, I I Baskin, V A Palyulin, N S Zefirov.   

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Year:  2003        PMID： 12856409     DOI： 10.1023/a:1023623803790

Source DB:  PubMed          Journal:  Dokl Biochem Biophys        ISSN： 1607-6729            Impact factor:   0.788


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  8 in total

1.  Mechanisms for activation and antagonism of an AMPA-sensitive glutamate receptor: crystal structures of the GluR2 ligand binding core.

Authors:  N Armstrong; E Gouaux
Journal:  Neuron       Date:  2000-10       Impact factor: 17.173

2.  Mutations in a putative agonist binding region of the AMPA-selective glutamate receptor channel.

Authors:  S Uchino; K Sakimura; K Nagahari; M Mishina
Journal:  FEBS Lett       Date:  1992-08-24       Impact factor: 4.124

3.  Comparative molecular field analysis (CoMFA). 1. Effect of shape on binding of steroids to carrier proteins.

Authors:  R D Cramer; D E Patterson; J D Bunce
Journal:  J Am Chem Soc       Date:  1988-08-01       Impact factor: 15.419

4.  8-(1H-imidazol-1-yl)-7-nitro-4(5H)-imidazo[1,2-alpha]quinoxalinone and related compounds: synthesis and structure-activity relationships for the AMPA-type non-NMDA receptor.

Authors:  J Ohmori; M Shimizu-Sasamata; M Okada; S Sakamoto
Journal:  J Med Chem       Date:  1997-06-20       Impact factor: 7.446

Review 5.  Neuropharmacology of AMPA and kainate receptors.

Authors:  D Bleakman; D Lodge
Journal:  Neuropharmacology       Date:  1998 Oct-Nov       Impact factor: 5.250

6.  Molecular similarity indices in a comparative analysis (CoMSIA) of drug molecules to correlate and predict their biological activity.

Authors:  G Klebe; U Abraham; T Mietzner
Journal:  J Med Chem       Date:  1994-11-25       Impact factor: 7.446

7.  Synthesis, ionotropic glutamate receptor binding affinity, and structure-activity relationships of a new set of 4,5-dihydro-8-heteroaryl-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylates analogues of TQX-173.

Authors:  D Catarzi; V Colotta; F Varano; G Filacchioni; A Galli; C Costagli; V Carlà
Journal:  J Med Chem       Date:  2001-09-13       Impact factor: 7.446

8.  Novel AMPA receptor antagonists: synthesis and structure-activity relationships of 1-hydroxy-7-(1H-imidazol-1-yl)-6-nitro-2,3(1H,4H)- quinoxalinedione and related compounds.

Authors:  J Ohmori; M Shimizu-Sasamata; M Okada; S Sakamoto
Journal:  J Med Chem       Date:  1996-09-27       Impact factor: 7.446
  8 in total

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