Literature DB >> 12819518

Suppression of cerebrospinal fluid HIV burden in antiretroviral naive patients on a potent four-drug antiretroviral regimen.

Michael A Polis1, Daniel L Suzman, Christian P Yoder, Jean M Shen, JoAnn M Mican, Robin L Dewar, Julia A Metcalf, Judith Falloon, Richard T Davey, Joseph A Kovacs, Mark B Feinberg, Henry Masur, Stephen C Piscitelli.   

Abstract

OBJECTIVE: To determine the longitudinal response of HIV in the cerebrospinal fluid (CSF) to highly active antiretroviral therapy (HAART) and to investigate the levels of indinavir penetrating into the CSF.
DESIGN: Open study of HIV-infected subjects naive to therapy with protease inhibitors.
SETTING: Tertiary care referral center.
SUBJECTS: Twenty-five participants were begun on indinavir, nevirapine, zidovudine, and lamivudine.
INTERVENTIONS: Lumbar punctures were performed prior to therapy and 2 and 6 months after beginning therapy. Plasma and CSF were assayed for routine cell counts, chemistries, HIV load and indinavir levels.
RESULTS: Twenty-two subjects had CSF HIV RNA level data available at all three time points, three others at baseline and 2 months. At month 2 of therapy, nine of 25 (36%) subjects had CSF HIV RNA levels > 50 HIV RNA copies/ml. By 6 months, all 22 subjects had CSF HIV RNA levels < 50 HIV RNA copies/ml. CSF white blood cell counts fell from a baseline mean of 5.3 x 10(6)/l to 1.9 x 10(6)/l (P = 0.013) at 6 months. Plasma indinavir levels declined rapidly while CSF levels remained stable throughout the 8-h dosing interval. The median CSF indinavir level was 71 ng/ml, approximating the upper limit of the 95% inhibitory concentration for indinavir against HIV-1.
CONCLUSIONS: CSF HIV RNA levels cannot be expected to fall below 50 HIV RNA copies/ml even after 2 months of therapy on HAART. Prolonged therapy may be required to suppress HIV levels within the central nervous system.

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Year:  2003        PMID: 12819518     DOI: 10.1097/00002030-200305230-00008

Source DB:  PubMed          Journal:  AIDS        ISSN: 0269-9370            Impact factor:   4.177


  12 in total

1.  Central nervous system penetration of antiretroviral drugs: pharmacokinetic, pharmacodynamic and pharmacogenomic considerations.

Authors:  Eric H Decloedt; Bernd Rosenkranz; Gary Maartens; John Joska
Journal:  Clin Pharmacokinet       Date:  2015-06       Impact factor: 6.447

Review 2.  CSF penetration by antiretroviral drugs.

Authors:  Christine Eisfeld; Doris Reichelt; Stefan Evers; Ingo Husstedt
Journal:  CNS Drugs       Date:  2013-01       Impact factor: 5.749

3.  The cerebrospinal fluid HIV risk score for assessing central nervous system activity in persons with HIV.

Authors:  Edward R Hammond; Rosa M Crum; Glenn J Treisman; Shruti H Mehta; Christina M Marra; David B Clifford; Susan Morgello; David M Simpson; Benjamin B Gelman; Ronald J Ellis; Igor Grant; Scott L Letendre; Justin C McArthur
Journal:  Am J Epidemiol       Date:  2014-06-24       Impact factor: 4.897

Review 4.  Antiretroviral therapy and central nervous system HIV type 1 infection.

Authors:  Richard W Price; Serena Spudich
Journal:  J Infect Dis       Date:  2008-05-15       Impact factor: 5.226

5.  Antiretroviral treatment effect on immune activation reduces cerebrospinal fluid HIV-1 infection.

Authors:  Elizabeth Sinclair; Rollie Ronquillo; Nicole Lollo; Steven G Deeks; Peter Hunt; Constantin T Yiannoutsos; Serena Spudich; Richard W Price
Journal:  J Acquir Immune Defic Syndr       Date:  2008-04-15       Impact factor: 3.731

6.  Darunavir concentrations in cerebrospinal fluid and blood in HIV-1-infected individuals.

Authors:  Aylin Yilmaz; Arash Izadkhashti; Richard W Price; Patrick W Mallon; Marc De Meulder; Philip Timmerman; Magnus Gisslén
Journal:  AIDS Res Hum Retroviruses       Date:  2009-04       Impact factor: 2.205

Review 7.  Should antiretroviral therapy for HIV infection be tailored for intracerebral penetration?

Authors:  P P Koopmans; R Ellis; B M Best; S Letendre
Journal:  Neth J Med       Date:  2009-06       Impact factor: 1.422

Review 8.  How much do antiretroviral drugs penetrate into the central nervous system?

Authors:  L Ene; D Duiculescu; S M Ruta
Journal:  J Med Life       Date:  2011-11-24

9.  Cerebrospinal fluid HIV infection and pleocytosis: relation to systemic infection and antiretroviral treatment.

Authors:  Serena S Spudich; Annelie C Nilsson; Nicole D Lollo; Teri J Liegler; Christos J Petropoulos; Steven G Deeks; Ellen E Paxinos; Richard W Price
Journal:  BMC Infect Dis       Date:  2005-11-02       Impact factor: 3.090

10.  Virological Response in Cerebrospinal Fluid to Antiretroviral Therapy in a Large Italian Cohort of HIV-Infected Patients with Neurological Disorders.

Authors:  Maria Letizia Giancola; Patrizia Lorenzini; Antonella Cingolani; Francesco Baldini; Simona Bossolasco; Teresa Bini; Laura Monno; Giovanna Picchi; Antonella d'Arminio Monforte; Paola Cinque; Valerio Tozzi; Andrea Antinori
Journal:  AIDS Res Treat       Date:  2012-08-26
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