Literature DB >> 12729674

Synthesis, anticholinesterase activity and structure-activity relationships of m-Aminobenzoic acid derivatives.

José Trujillo-Ferrara1, Leticia Montoya Cano, Michel Espinoza-Fonseca.   

Abstract

The synthesis, acetylcholinesterase inhibitory capacity and structure-activity relationships of simple-structured m-Aminobenzoic acid derivatives are reported. Compound 1b was found to be more potent than galanthamine and tacrine in inhibiting acetylcholinesterase.

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Year:  2003        PMID： 12729674     DOI： 10.1016/s0960-894x(03)00198-7

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  3 in total

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Authors:  Ashwani Kumar; Sandeep Jain; Milind Parle; Neelam Jain; Parvin Kumar
Journal:  EXCLI J       Date:  2013-12-13       Impact factor: 4.068
  3 in total

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