Literature DB >> 12540230

5-HT4 receptor ligands: applications and new prospects.

Michel Langlois1, Rodolphe Fischmeister.   

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Year:  2003        PMID: 12540230     DOI: 10.1021/jm020099f

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  22 in total

1.  Functional studies of the 5'-untranslated region of human 5-HT4 receptor mRNA.

Authors:  Marjorie Maillet; Monique Gastineau; Pascal Bochet; Marie-Liesse Asselin-Labat; Eric Morel; Jean-Noël Laverrière; Anne-Marie Lompré; Rodolphe Fischmeister; Frank Lezoualc'h
Journal:  Biochem J       Date:  2005-04-15       Impact factor: 3.857

2.  Selective desensitization of the 5-HT4 receptor-mediated response in pig atrium but not in stomach.

Authors:  J H De Maeyer; J A J Schuurkes; R A Lefebvre
Journal:  Br J Pharmacol       Date:  2009-01-13       Impact factor: 8.739

3.  Multivalent ligands for the serotonin 5-HT4 receptor.

Authors:  Federica Castriconi; Marco Paolino; Alessandro Donati; Germano Giuliani; Maurizio Anzini; Laura Mennuni; Chiara Sabatini; Marco Lanza; Gianfranco Caselli; Francesco Makovec; Maria Sbraccia; Paola Molinari; Tommaso Costa; Andrea Cappelli
Journal:  Medchemcomm       Date:  2017-02-09       Impact factor: 3.597

4.  Differences between the abilities of tegaserod and motilin receptor agonists to stimulate gastric motility in vitro.

Authors:  E M Jarvie; V J North Laidler; S Corcoran; A Bassil; G J Sanger
Journal:  Br J Pharmacol       Date:  2007-01-08       Impact factor: 8.739

5.  Cardiovascular effects of cisapride and prucalopride on human 5-HT4 receptors in transgenic mice.

Authors:  Nicolas Keller; Stefan Dhein; Joachim Neumann; Ulrich Gergs
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2018-06-09       Impact factor: 3.000

6.  Prucalopride is a partial agonist through human and porcine atrial 5-HT4 receptors: comparison with recombinant human 5-HT4 splice variants.

Authors:  Kurt A Krobert; Trond Brattelid; Finn Olav Levy; Alberto J Kaumann
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2005-07-13       Impact factor: 3.000

7.  Visceral analgesic effect of 5-HT(4) receptor agonist in rats involves the rostroventral medulla (RVM).

Authors:  Jyoti N Sengupta; Aaron Mickle; Pradeep Kannampalli; Russell Spruell; John McRorie; Reza Shaker; Adrian Miranda
Journal:  Neuropharmacology       Date:  2013-12-12       Impact factor: 5.250

8.  Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography.

Authors:  Rong Xu; Jinsoo Hong; Cheryl L Morse; Victor W Pike
Journal:  J Med Chem       Date:  2010-10-14       Impact factor: 7.446

9.  Development of subnanomolar-affinity serotonin 5-HT4 receptor ligands based on quinoline structures.

Authors:  Federica Castriconi; Marco Paolino; Giorgio Grisci; Cinzia Maria Francini; Annalisa Reale; Germano Giuliani; Maurizio Anzini; Gianluca Giorgi; Laura Mennuni; Chiara Sabatini; Marco Lanza; Gianfranco Caselli; Andrea Cappelli
Journal:  Medchemcomm       Date:  2018-07-03       Impact factor: 3.597

10.  New insights into the human 5-HT4 receptor binding site: exploration of a hydrophobic pocket.

Authors:  Lucie Rivail; Mireille Giner; Monique Gastineau; Magali Berthouze; Jean-Louis Soulier; Rodolphe Fischmeister; Frank Lezoualc'h; Bernard Maigret; Sames Sicsic; Isabelle Berque-Bestel
Journal:  Br J Pharmacol       Date:  2004-09-06       Impact factor: 8.739

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