Literature DB >> 12491396

The total synthesis of proteasome inhibitors TMC-95A and TMC-95B: discovery of a new method to generate cis-propenyl amides.

Songnian Lin1, Samuel J Danishefsky.   

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Year:  2002        PMID： 12491396     DOI： 10.1002/1521-3773(20020201)41:3<512::aid-anie512>3.0.co;2-r

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


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  7 in total

1.  A concise, total synthesis of the TMC-95A/B proteasome inhibitors.

Authors:  Brian K Albrecht; Robert M Williams
Journal:  Proc Natl Acad Sci U S A       Date:  2004-05-26       Impact factor: 11.205

2.  Total synthesis of enantiopure phalarine via a stereospecific Pictet-Spengler reaction: traceless transfer of chirality from L-tryptophan.

Authors:  John D Trzupek; Dongjoo Lee; Brendan M Crowley; Vasilios M Marathias; Samuel J Danishefsky
Journal:  J Am Chem Soc       Date:  2010-06-23       Impact factor: 15.419

3.  Total synthesis of TMC-95A and -B via a new reaction leading to Z-enamides. Some preliminary findings as to SAR.

Authors:  Songnian Lin; Zhi-Qiang Yang; Benjamin H B Kwok; Michael Koldobskiy; Craig M Crews; Samuel J Danishefsky
Journal:  J Am Chem Soc       Date:  2004-05-26       Impact factor: 15.419

4.  Sequential Functionalization of meta-C-H and ipso-C-O Bonds of Phenols.

Authors:  Jiancong Xu; Jingjing Chen; Feng Gao; Shuguang Xie; Xiaohua Xu; Zhong Jin; Jin-Quan Yu
Journal:  J Am Chem Soc       Date:  2019-01-24       Impact factor: 15.419

5.  Stereospecific Ring Contraction of Bromocycloheptenes through Dyotropic Rearrangements via Nonclassical Carbocation-Anion Pairs.

Authors:  Shermin S Goh; Pier Alexandre Champagne; Sureshbabu Guduguntla; Takashi Kikuchi; Makoto Fujita; K N Houk; Ben L Feringa
Journal:  J Am Chem Soc       Date:  2018-04-05       Impact factor: 15.419

6.  Natural product scaffolds as inspiration for the design and synthesis of 20S human proteasome inhibitors.

Authors:  Grace E Hubbell; Jetze J Tepe
Journal:  RSC Chem Biol       Date:  2020-09-16

7.  Peptide and Peptide-Like Modulators of 20S Proteasome Enzymatic Activity in Cancer Cells.

Authors:  Carlos García-Echeverría
Journal:  Int J Pept Res Ther       Date:  2006-03-04       Impact factor: 1.931
  7 in total

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