Literature DB >> 12490852

Activation of the ras/raf-1 signal transduction pathway in carcinoid tumor cells results in morphologic transdifferentiation.

Rebecca S Sippel1, Herbert Chen.   

Abstract

BACKGROUND: Recent studies of neuroendocrine tumor cell lines suggest that ras/raf-1 activation could be detrimental to tumorigenesis. The mechanism by which it alters neuroendocrine tumor cells is unclear. We hypothesize that activation of the ras/raf signal transduction pathway may alter gastrointestinal carcinoid cells by inducing morphologic transdifferentiation.
METHODS: Pancreatic carcinoid (BON) cells were transduced in a stable manner with an estrogen inducible raf-1 fusion protein (creating "BON-raf cells"). BON and BON-raf cells were then treated with either control or 1 micromol/L estradiol (E2). Western blots were used to confirm the phosphorylation of extracellular signal-regulated kinase 1/2. Morphologic changes were evaluated using light and electron microscopy.
RESULTS: Western blots using antibodies against phosphorylated and unphosphorylated extracellular signal-regulated kinase 1/2. confirmed that phosphorylation was only present in the BON-raf E2 cells. BON cells treated with control and E2 and BON-raf cells treated with control all looked identical in culture. After treatment with E2 to induce raf-1, the BON-raf cells underwent dramatic morphologic changes. Under light and electron microscopy the cells became flatter and developed much sharper cellular borders mimicking cellular differentiation.
CONCLUSIONS: Activation of the ras/raf-1 signal transduction pathway leads to prominent phenotypic changes that resemble differentiation of gastrointestinal carcinoid cells in vitro.

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Year:  2002        PMID: 12490852     DOI: 10.1067/msy.2002.128877

Source DB:  PubMed          Journal:  Surgery        ISSN: 0039-6060            Impact factor:   3.982


  10 in total

Review 1.  Therapeutic and palliative options for diffuse neuroendocrine metastatic disease.

Authors:  Kyle Holen
Journal:  J Gastrointest Surg       Date:  2006-03       Impact factor: 3.452

Review 2.  Signaling mechanisms in neuroendocrine tumors as targets for therapy.

Authors:  Barbara Zarebczan; Herbert Chen
Journal:  Endocrinol Metab Clin North Am       Date:  2010-12       Impact factor: 4.741

3.  Overexpression of Raf-1 and ERK1/2 in sacral chordoma and association with tumor recurrence.

Authors:  Kai Zhang; Hao Chen; Bin Zhang; Jiajia Sun; Jian Lu; Kangwu Chen; Huilin Yang
Journal:  Int J Clin Exp Pathol       Date:  2015-01-01

Review 4.  Signaling pathways as specific pharmacologic targets for neuroendocrine tumor therapy: RET, PI3K, MEK, growth factors, and Notch.

Authors:  Yvette Carter; Renata Jaskula-Sztul; Herbert Chen; Haggi Mazeh
Journal:  Neuroendocrinology       Date:  2012-02-14       Impact factor: 4.914

5.  Interaction of BAG1 and Hsp70 mediates neuroprotectivity and increases chaperone activity.

Authors:  Jan Liman; Sundar Ganesan; Christoph P Dohm; Stan Krajewski; John C Reed; Mathias Bähr; Fred S Wouters; Pawel Kermer
Journal:  Mol Cell Biol       Date:  2005-05       Impact factor: 4.272

6.  Combined blockade of signalling pathways shows marked anti-tumour potential in phaeochromocytoma cell lines.

Authors:  Svenja Nölting; Edwin Garcia; Ghassan Alusi; Alessio Giubellino; Karel Pacak; Márta Korbonits; Ashley B Grossman
Journal:  J Mol Endocrinol       Date:  2012-07-25       Impact factor: 5.098

7.  Focal adhesion kinase, a downstream mediator of Raf-1 signaling, suppresses cellular adhesion, migration, and neuroendocrine markers in BON carcinoid cells.

Authors:  Li Ning; Herbert Chen; Muthusamy Kunnimalaiyaan
Journal:  Mol Cancer Res       Date:  2010-04-20       Impact factor: 5.852

8.  Raf-1 activation in gastrointestinal carcinoid cells decreases tumor cell adhesion.

Authors:  David Yü Greenblatt; Muthusamy Kunnimalaiyaan; Herbert Chen
Journal:  Am J Surg       Date:  2007-03       Impact factor: 2.565

9.  ZM336372, a Raf-1 activator, causes suppression of proliferation in a human hepatocellular carcinoma cell line.

Authors:  Dustin Deming; Peter Geiger; Herbert Chen; Abram Vaccaro; Muthusamy Kunnimalaiyaan; Kyle Holen
Journal:  J Gastrointest Surg       Date:  2008-05       Impact factor: 3.452

Review 10.  PI3K-AKT-mTOR-signaling and beyond: the complex network in gastroenteropancreatic neuroendocrine neoplasms.

Authors:  Franziska Briest; Patricia Grabowski
Journal:  Theranostics       Date:  2014-01-29       Impact factor: 11.556

  10 in total

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