| Literature DB >> 12182666 |
Zhongxing Zhang1, Zhong Yang, Henry Wong, Juliang Zhu, Nicholas A Meanwell, John F Kadow, Tao Wang.
Abstract
Conditions for attachment of acetyl chloride, benzoyl chloride, and chloromethyl oxalate to the 3-position of 4-, 5-, 6-, or 7-azaindoles were explored. Best results were achieved with an excess of AlCl(3) in CH(2)Cl(2) followed by the addition of an acyl chloride at room temperature.Entities:
Year: 2002 PMID： 12182666 DOI： 10.1021/jo020135i
Source DB: PubMed Journal: J Org Chem ISSN： 0022-3263 Impact factor: 4.354