Literature DB >> 12094204

A novel mechanism for the beneficial vascular effects of high-density lipoprotein cholesterol: enhanced vasorelaxation and increased endothelial nitric oxide synthase expression.

Jeffrey T Kuvin1, Maria E Rämet, Ayan R Patel, Natesa G Pandian, Michael E Mendelsohn, Richard H Karas.   

Abstract

BACKGROUND: Low levels of high-density lipoprotein (HDL) cholesterol increase the risk of coronary artery disease (CAD), and recent clinical studies suggest that interventions in low-HDL patients are beneficial. The purpose of this study was to examine the effect of increased HDL levels on endothelium-dependent vasodilation.
METHODS: We studied patients with CAD with a low-density lipoprotein (LDL) level of <100 mg/dL. Patients with an HDL level of < or =36 mg/dL were treated with niacin (n = 11), and patients with an HDL level of >36 mg/dL were followed as controls (n = 10). Baseline and 3-month follow-up studies of flow-mediated dilation (FMD) and blood lipid levels were obtained.
RESULTS: HDL levels increased from 30.1 +/- 1.2 to 40.5 +/- 1.2 mg/dL in the niacin-treated patients (P <.001) but remained unchanged in the control patients. At baseline, FMD was impaired in both the treated (6.5% +/- 1%) and the control (7.3% +/- 1%) patients compared with 10 healthy subjects (16% +/- 2%, P <.01). After 3 months, FMD improved in the niacin-treated patients (11.8% +/- 1%, P =.001) but remained unchanged in the control patients (6.2% +/- 1%). Exposure of cultured human vascular endothelial cells to HDL in vitro enhanced expression of endothelial nitric oxide synthase (eNOS), as shown by immunoblotting.
CONCLUSIONS: In patients with CAD and well-controlled LDL levels, elevation of HDL with niacin improves endothelial function. HDL increases eNOS protein expression in cultured vascular endothelial cells. Taken together, these observations suggest that HDL-mediated increases in eNOS expression may contribute to the observed enhancement in vasorelaxation and thus support a previously unrecognized mechanism for the beneficial cardiovascular effects of HDL.

Entities:  

Mesh:

Substances:

Year:  2002        PMID: 12094204     DOI: 10.1067/mhj.2002.123145

Source DB:  PubMed          Journal:  Am Heart J        ISSN: 0002-8703            Impact factor:   4.749


  42 in total

1.  HDL action on the vascular wall: is the answer NO?

Authors:  Philip W Shaul; Chieko Mineo
Journal:  J Clin Invest       Date:  2004-02       Impact factor: 14.808

Review 2.  Mechanisms, significance and treatment of vascular dysfunction in type 2 diabetes mellitus: focus on lipid-regulating therapy.

Authors:  Richard J Woodman; Gerard T Chew; Gerald F Watts
Journal:  Drugs       Date:  2005       Impact factor: 9.546

Review 3.  Beyond high-density lipoprotein cholesterol levels evaluating high-density lipoprotein function as influenced by novel therapeutic approaches.

Authors:  Emil M deGoma; Rolando L deGoma; Daniel J Rader
Journal:  J Am Coll Cardiol       Date:  2008-06-10       Impact factor: 24.094

Review 4.  High density lipoproteins and endothelial functions: mechanistic insights and alterations in cardiovascular disease.

Authors:  Meliana Riwanto; Ulf Landmesser
Journal:  J Lipid Res       Date:  2013-07-20       Impact factor: 5.922

5.  Extended-Release Niacin Versus Fenofibrate in HIV-Infected Participants With Low High-Density Lipoprotein Cholesterol: Effects on Endothelial Function, Lipoproteins, and Inflammation.

Authors:  Michael P Dubé; Lauren Komarow; Carl J Fichtenbaum; Joseph J Cadden; Edgar T Overton; Howard N Hodis; Judith S Currier; James H Stein
Journal:  Clin Infect Dis       Date:  2015-05-15       Impact factor: 9.079

6.  Associations of cardiovascular risk factors with two surrogate markers of subclinical atherosclerosis: endothelial function and carotid intima media thickness.

Authors:  Kathleen V Fitch; Eleni Stavrou; Sara E Looby; Linda Hemphill; Michael R Jaff; Steven K Grinspoon
Journal:  Atherosclerosis       Date:  2011-04-16       Impact factor: 5.162

Review 7.  A "hot" topic in dyslipidemia management--"how to beat a flush": optimizing niacin tolerability to promote long-term treatment adherence and coronary disease prevention.

Authors:  Terry A Jacobson
Journal:  Mayo Clin Proc       Date:  2010-04       Impact factor: 7.616

8.  Novel small molecule therapeutics for sickle cell disease: nitric oxide, carbon monoxide, nitrite, and apolipoprotein A-I.

Authors:  Gregory J Kato
Journal:  Hematology Am Soc Hematol Educ Program       Date:  2008

9.  Extended-release niacin/laropiprant improves endothelial function in patients after myocardial infarction.

Authors:  Urska Bregar; Borut Jug; Irena Keber; Matija Cevc; Miran Sebestjen
Journal:  Heart Vessels       Date:  2013-05-28       Impact factor: 2.037

10.  ABCG1 and HDL protect against endothelial dysfunction in mice fed a high-cholesterol diet.

Authors:  Naoki Terasaka; Shuiqing Yu; Laurent Yvan-Charvet; Nan Wang; Nino Mzhavia; Read Langlois; Tamara Pagler; Rong Li; Carrie L Welch; Ira J Goldberg; Alan R Tall
Journal:  J Clin Invest       Date:  2008-10-16       Impact factor: 14.808

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.