Literature DB >> 12067541

Antimalarial activities of ring-substituted bioimidazoles.

Rahul Jain1, Suryanarayana Vangapandu, Meenakshi Jain, Navneet Kaur, Savita Singh, Prati Pal Singh.   

Abstract

We report in vitro antimalarial activities against chloroquine sensitive and resistant Plasmodium falciparum strains, and in vivo activities against Plasmodium berghei in mice for four series of ring-substituted-L-histidines and histamines.

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Year:  2002        PMID: 12067541     DOI: 10.1016/s0960-894x(02)00289-5

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN: 0960-894X            Impact factor:   2.823


  2 in total

1.  2-tert-butyl-8-quinolinamines exhibit potent blood schizontocidal antimalarial activity via inhibition of heme crystallization.

Authors:  Nguyen Tien Huy; Keisuke Mizunuma; Kirandeep Kaur; Nguyen Thanh Thuy Nhien; Meenakshi Jain; Dinh Thanh Uyen; Shigeharu Harada; Rahul Jain; Kaeko Kamei
Journal:  Antimicrob Agents Chemother       Date:  2007-06-11       Impact factor: 5.191

Review 2.  An epigrammatic status of the 'azole'-based antimalarial drugs.

Authors:  Mousmee Sharma; Parteek Prasher
Journal:  RSC Med Chem       Date:  2019-12-23
  2 in total

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