Literature DB >> 11988746

Amyloid-lowering isocoumarins are not direct inhibitors of gamma-secretase.

William P Esler, Chittaranjan Das, William A Campbell, W Taylor Kimberly, Anna Y Kornilova, Thekla S Diehl, Wenjuan Ye, Beth L Ostaszewski, Weiming Xia, Dennis J Selkoe, Michael S Wolfe.   

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Year:  2002        PMID: 11988746     DOI: 10.1038/ncb0502-e110b

Source DB:  PubMed          Journal:  Nat Cell Biol        ISSN: 1465-7392            Impact factor:   28.824


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  6 in total

1.  Electron microscopic structure of purified, active gamma-secretase reveals an aqueous intramembrane chamber and two pores.

Authors:  Vlado K Lazarov; Patrick C Fraering; Wenjuan Ye; Michael S Wolfe; Dennis J Selkoe; Huilin Li
Journal:  Proc Natl Acad Sci U S A       Date:  2006-04-24       Impact factor: 11.205

2.  Presenilins mediate a dual intramembranous gamma-secretase cleavage of Notch-1.

Authors:  Masayasu Okochi; Harald Steiner; Akio Fukumori; Hisashi Tanii; Taisuke Tomita; Toshihisa Tanaka; Takeshi Iwatsubo; Takashi Kudo; Masatoshi Takeda; Christian Haass
Journal:  EMBO J       Date:  2002-10-15       Impact factor: 11.598

Review 3.  Inhibition of gamma-secretase as a therapeutic intervention for Alzheimer's disease: prospects, limitations and strategies.

Authors:  Geneviève Evin; Marijke Fleur Sernee; Colin L Masters
Journal:  CNS Drugs       Date:  2006       Impact factor: 5.749

4.  Alzheimer's disease-linked presenilin mutation (PS1M146L) induces filamin expression and γ-secretase independent redistribution.

Authors:  Qun Lu; Kai Ding; Matthew P Frosch; Shiloh Jones; Michael Wolfe; Weiming Xia; George W Lanford
Journal:  J Alzheimers Dis       Date:  2010       Impact factor: 4.472

Review 5.  BACE and gamma-secretase characterization and their sorting as therapeutic targets to reduce amyloidogenesis.

Authors:  Neville Marks; Martin J Berg
Journal:  Neurochem Res       Date:  2009-09-17       Impact factor: 3.996

Review 6.  Gamma-secretase inhibition and modulation for Alzheimer's disease.

Authors:  Michael S Wolfe
Journal:  Curr Alzheimer Res       Date:  2008-04       Impact factor: 3.498

  6 in total

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