Literature DB >> 11933229

Vancomycin resistance: small molecule approaches targeting the bacterial cell wall biosynthesis.

Roderich D Süssmuth1.   

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Year:  2002        PMID： 11933229     DOI： 10.1002/1439-7633(20020402)3:4<295::AID-CBIC295>3.0.CO;2-G

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  10 in total

1.  N-Terminus Alkylation of Vancomycin: Ligand Binding Affinity, Antimicrobial Activity, and Site-Specific Nature of Quaternary Trimethylammonium Salt Modification.

Authors:  Zhi-Chen Wu; Nicholas A Isley; Dale L Boger
Journal:  ACS Infect Dis       Date:  2018-08-08       Impact factor: 5.084

2.  Total syntheses and initial evaluation of [Ψ[C(═S)NH]Tpg⁴]vancomycin, [Ψ[C(═NH)NH]Tpg⁴]vancomycin, [Ψ[CH₂NH]Tpg⁴]vancomycin, and their (4-chlorobiphenyl)methyl derivatives: synergistic binding pocket and peripheral modifications for the glycopeptide antibiotics.

Authors:  Akinori Okano; Atsushi Nakayama; Kejia Wu; Erick A Lindsey; Alex W Schammel; Yiqing Feng; Karen C Collins; Dale L Boger
Journal:  J Am Chem Soc       Date:  2015-03-09       Impact factor: 15.419

3.  Total synthesis of [Ψ[C(═S)NH]Tpg4]vancomycin aglycon, [Ψ[C(═NH)NH]Tpg4]vancomycin aglycon, and related key compounds: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding.

Authors:  Jian Xie; Akinori Okano; Joshua G Pierce; Robert C James; Simon Stamm; Christine M Crane; Dale L Boger
Journal:  J Am Chem Soc       Date:  2012-01-06       Impact factor: 15.419

4.  Total synthesis and evaluation of [Psi[CH2NH]Tpg4]vancomycin aglycon: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding.

Authors:  Brendan M Crowley; Dale L Boger
Journal:  J Am Chem Soc       Date:  2006-03-08       Impact factor: 15.419

5.  Synthesis and evaluation of selected key methyl ether derivatives of vancomycin aglycon.

Authors:  Christine M Crane; Joshua G Pierce; Siegfried S F Leung; Julian Tirado-Rives; William L Jorgensen; Dale L Boger
Journal:  J Med Chem       Date:  2010-10-14       Impact factor: 7.446

6.  Probing the role of the vancomycin e-ring aryl chloride: selective divergent synthesis and evaluation of alternatively substituted E-ring analogues.

Authors:  Joseph R Pinchman; Dale L Boger
Journal:  J Med Chem       Date:  2013-05-13       Impact factor: 7.446

7.  Synthesis and binding studies of two new macrocyclic receptors for the stereoselective recognition of dipeptides.

Authors:  Ana Maria Castilla; M Morgan Conn; Pablo Ballester
Journal:  Beilstein J Org Chem       Date:  2010-01-19       Impact factor: 2.883

8.  Synthesis and evaluation of vancomycin aglycon analogues that bear modifications in the N-terminal D-leucyl amino acid.

Authors:  Christine M Crane; Dale L Boger
Journal:  J Med Chem       Date:  2009-03-12       Impact factor: 7.446

9.  Silver(I)-promoted conversion of thioamides to amidines: divergent synthesis of a key series of vancomycin aglycon residue 4 amidines that clarify binding behavior to model ligands.

Authors:  Akinori Okano; Robert C James; Joshua G Pierce; Jian Xie; Dale L Boger
Journal:  J Am Chem Soc       Date:  2012-05-17       Impact factor: 15.419

10.  Total synthesis of [Ψ[C(═NH)NH]Tpg(4)]vancomycin and its (4-chlorobiphenyl)methyl derivative: impact of peripheral modifications on vancomycin analogues redesigned for dual D-Ala-D-Ala and D-Ala-D-Lac binding.

Authors:  Akinori Okano; Atsushi Nakayama; Alex W Schammel; Dale L Boger
Journal:  J Am Chem Soc       Date:  2014-09-16       Impact factor: 15.419
  10 in total

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