Literature DB >> 11914204

Vitreous penetration of levofloxacin in the uninflamed phakic human eye.

E N Herbert1, I A Pearce, J McGalliard, D Wong, C Groenewald.   

Abstract

AIMS: To assess the vitreous penetration of oral levofloxacin (a new fluoroquinolone antibiotic with improved Gram positive activity) in uninflamed phakic eyes.
METHODS: 15 patients for macula hole surgery were recruited to the study. 10 received a single 500 mg dose of levofloxacin by mouth preoperatively. Five acted as controls. Serum and undiluted vitreous samples were obtained at surgery and analysed by HPLC.
RESULTS: Levofloxacin was detectable 2.5 hours after administration in the vitreous. A peak concentration of 1.6 microg/ml (or mg/l) was measured between 2.5 and 4 hours post-dose.
CONCLUSION: Oral levofloxacin reaches the vitreous rapidly in the uninflamed phakic eye. Levels did not reach MIC(90) for the commonest infecting organisms. Nevertheless, levofloxacin would be expected to be active against a higher proportion of infecting organisms than either ciprofloxacin or ofloxacin.

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Year:  2002        PMID: 11914204      PMCID: PMC1771086          DOI: 10.1136/bjo.86.4.387

Source DB:  PubMed          Journal:  Br J Ophthalmol        ISSN: 0007-1161            Impact factor:   4.638


  13 in total

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Authors:  R G Fiscella; T K Nguyen; M J Cwik; B A Phillpotts; S M Friedlander; D C Alter; M J Shapiro; N P Blair; J P Gieser
Journal:  Ophthalmology       Date:  1999-12       Impact factor: 12.079

2.  The intravitreal penetration of orally administered ciprofloxacin in humans.

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3.  In-vitro activity of trovafloxacin against clinical bacterial isolates from patients with cancer.

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4.  Intracorneal, aqueous humor, and vitreous humor penetration of topical and oral ofloxacin.

Authors:  E D Donnenfeld; H D Perry; R W Snyder; R Moadel; M Elsky; H Jones
Journal:  Arch Ophthalmol       Date:  1997-02

5.  Intravitreal penetration of oral ciprofloxacin in humans.

Authors:  F Z el Baba; M D Trousdale; W J Gauderman; D G Wagner; P E Liggett
Journal:  Ophthalmology       Date:  1992-04       Impact factor: 12.079

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Journal:  Ophthalmology       Date:  1999-07       Impact factor: 12.079

7.  Intravitreal penetration of teicoplanin.

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Authors:  G Gatti; G Panozzo
Journal:  Antimicrob Agents Chemother       Date:  1995-02       Impact factor: 5.191

Review 9.  Levofloxacin. A review of its antibacterial activity, pharmacokinetics and therapeutic efficacy.

Authors:  R Davis; H M Bryson
Journal:  Drugs       Date:  1994-04       Impact factor: 9.546

10.  Results of the Endophthalmitis Vitrectomy Study. A randomized trial of immediate vitrectomy and of intravenous antibiotics for the treatment of postoperative bacterial endophthalmitis. Endophthalmitis Vitrectomy Study Group.

Authors: 
Journal:  Arch Ophthalmol       Date:  1995-12
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4.  Evaluation of the levofloxacin release characters from a rabbit foldable capsular vitreous body.

Authors:  Zhaoxin Jiang; Ting Wang; Biyan Pan; Zhiyong Xie; Peijuan Wang; Yaqin Liu; Qianying Gao
Journal:  Int J Nanomedicine       Date:  2011-12-30

5.  Risk Factors for Endophthalmitis Following Open Globe Injuries: A 17-Year Analysis.

Authors:  Asad F Durrani; Peter Y Zhao; Yunshu Zhou; Michael Huvard; Lyna Azzouz; Jason M Keil; Stephen T Armenti; Vaidehi S Dedania; David C Musch; David N Zacks
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