Literature DB >> 11731739

Growth inhibition of epidermal growth factor-stimulated human glioblastoma cells by nicardipine in vitro.

C Huang1, S Hu, B Chen.   

Abstract

BACKGROUND: The objective of this work was to observe and analyze the effects of epidermal growth factor (EGF) and the calcium channel antagonist nicardipine on the growth of U251MG, a human malignant glioma cell line, which have high-affinity EGF receptors.
METHODS: The growth effects of EGF and nicardipine on U251MG cultured in serum-free and serum-supplemented (10% fetal bovine serum, FBS) medium respectively were observed by MTT colorimeritric analysis.
RESULTS: EGF significantly enhanced the growth of U251MG cells in a dose-dependent manner in serum-free medium. The maximal effect was seen at 20 ng/ml. The effects of EGF approximated those obtained in 10% FBS. Nicardipine decreased U251MG cell proliferation, especially in serum-supplemented medium, and completely blocked the growth-stimulated effects of EGF. The combined effects of EGF (10 ng/ml) and nicardipine equaled those of nicardipine alone.
CONCLUSIONS: When serum was absent, the U251MG cells showed a pronounced mitogenic response to EGF in a dose-dependent manner, which approximated that achieved with 10% FBS. The addition of serum obscured this effect. Nicardipine suppressed the growth of U251MG cells and completely blocked the growth-stimulated effects of EGF may suggest a possible role of this drug as adjuvant therapy for human malignant gliomas.

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Year:  2001        PMID: 11731739

Source DB:  PubMed          Journal:  J Neurosurg Sci        ISSN: 0390-5616            Impact factor:   2.279


  2 in total

Review 1.  Receptor tyrosine kinase targeting in glioblastoma: performance, limitations and future approaches.

Authors:  Oana Alexandru; Cristina Horescu; Ani-Simona Sevastre; Catalina Elena Cioc; Carina Baloi; Alexandru Oprita; Anica Dricu
Journal:  Contemp Oncol (Pozn)       Date:  2020-03-30

2.  Nicardipine sensitizes temozolomide by inhibiting autophagy and promoting cell apoptosis in glioma stem cells.

Authors:  Jia Shi; Xuchen Dong; Haoran Li; Haiyang Wang; Qianqian Jiang; Liang Liu; Liping Wang; Jun Dong
Journal:  Aging (Albany NY)       Date:  2021-02-17       Impact factor: 5.682

  2 in total

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