Literature DB >> 11578236

Novel syntheses of 2,3-dihydro-1,5-benzothiazepin-4(5h)-ones and 2h-1,4-benzothiazin-3(4h)-ones.

A R Katritzky1, H H Odens, S Zhang, C J Rostek, O W Maender.   

Abstract

Nucleophilic additions of alpha-mercaptoalkanoate esters and beta-mercaptoalkanoate acids to benzoquinone diimines, followed by cyclization with trifluoroacetic acid or 1,3-dicyclohexylcarbodiimide (DCC), provide novel, high-yielding syntheses of 2H-1,4-benzothiazin-3(4H)-ones (3a-f) and 2,3-dihydro-1,5-benzothiazepin-4(5H)-ones (5a-c), respectively.

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Year:  2001        PMID: 11578236     DOI: 10.1021/jo0101959

Source DB:  PubMed          Journal:  J Org Chem        ISSN: 0022-3263            Impact factor:   4.354


  4 in total

1.  Parallel Synthesis of Structurally Diverse Aminobenzimidazole Tethered Sultams and Benzothiazepinones.

Authors:  Sureshbabu Dadiboyena; Adel Nefzi
Journal:  Tetrahedron Lett       Date:  2012-12-19       Impact factor: 2.415

2.  Scientia pharmaceutica, autorenhinweise 2013.

Authors: 
Journal:  Sci Pharm       Date:  2012-12-10

3.  [Not Available].

Authors: 
Journal:  Sci Pharm       Date:  2014-11-22

4.  [Not Available].

Authors: 
Journal:  Sci Pharm       Date:  2016-01-01
  4 in total

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