Literature DB >> 11505021

Relationship of brain ethanol metabolism to the hypnotic effect of ethanol. I: Studies in outbred animals.

S M Zimatkin1, A V Liopo, V S Slychenkov , R A Deitrich.   

Abstract

BACKGROUND: This study was designed to investigate the relationship between the ethanol-oxidizing capacity of the brain, accumulation of acetaldehyde, and ethanol-induced hypnosis in animals in vivo.
METHODS: Randomly outbred albino rats were treated with ethanol, and the duration of ethanol-induced loss of the righting response (sleep time) was measured. They were killed 2 weeks later (without further in vivo administration of ethanol), and brain homogenates were prepared to measure the accumulation of acetaldehyde from ethanol added in vitro. In a similar way, we determined the sleep time and, 5 days later, the rates of acetaldehyde accumulation in brains of heterogeneous mice.
RESULTS: Significant correlations between the duration of ethanol-induced sleep and acetaldehyde accumulation in vitro were found. The Km value of the process of acetaldehyde accumulation was lower in long-sleeping, as compared with short-sleeping, rats. A similar result was also obtained in genetically heterogeneous mice. Animals with a longer duration of ethanol-induced sleep had a higher level of the accumulation of ethanol-derived acetaldehyde in brain homogenates, as compared with the short-sleeping mice. Rats and mice with the intermediate duration of ethanol-induced sleep had an intermediate value of acetaldehyde accumulation in brain homogenates. There was no correlation between brain catalase activity and ethanol-induced loss of the righting response in either the rats or the mice.
CONCLUSIONS: This study is a direct demonstration of the positive correlation between ethanol-derived acetaldehyde accumulation in vitro in the brain and a central (behavioral) effect of alcohol in outbred rats and mice in vivo.

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Year:  2001        PMID: 11505021

Source DB:  PubMed          Journal:  Alcohol Clin Exp Res        ISSN: 0145-6008            Impact factor:   3.455


  6 in total

1.  Acetate-dependent mechanisms of inborn tolerance to ethanol.

Authors:  Sergey M Zimatkin; Nikolay A Oganesian; Yury V Kiselevski; Richard A Deitrich
Journal:  Alcohol Alcohol       Date:  2011-02-24       Impact factor: 2.826

2.  Binge ethanol administration enhances the MDMA-induced long-term 5-HT neurotoxicity in rat brain.

Authors:  María Izco; Laura Orio; Esther O'Shea; M Isabel Colado
Journal:  Psychopharmacology (Berl)       Date:  2006-10-18       Impact factor: 4.530

3.  Reward and relapse: complete gene-induced dissociation in an animal model of alcohol dependence.

Authors:  María E Quintanilla; Lutske Tampier; Eduardo Karahanian; Mario Rivera-Meza; Mario Herrera-Marschitz; Yedy Israel
Journal:  Alcohol Clin Exp Res       Date:  2011-09-06       Impact factor: 3.455

4.  Oxidation of ethanol in the rat brain and effects associated with chronic ethanol exposure.

Authors:  Jie Wang; Hongying Du; Lihong Jiang; Xiaoxian Ma; Robin A de Graaf; Kevin L Behar; Graeme F Mason
Journal:  Proc Natl Acad Sci U S A       Date:  2013-08-12       Impact factor: 11.205

5.  Behavioral characterization of acetaldehyde in C57BL/6J mice: locomotor, hypnotic, anxiolytic and amnesic effects.

Authors:  Etienne Quertemont; Sophie Tambour; Pascale Bernaerts; Sergey M Zimatkin; Ezio Tirelli
Journal:  Psychopharmacology (Berl)       Date:  2004-05-25       Impact factor: 4.530

6.  Alcohol ADME in primates studied with positron emission tomography.

Authors:  Zizhong Li; Youwen Xu; Don Warner; Nora D Volkow
Journal:  PLoS One       Date:  2012-10-01       Impact factor: 3.240

  6 in total

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