Literature DB >> 11504648

Synthesis and pharmacological activity of metabolites of the 5-HT(4) receptor antagonist SB-207266.

M Fedouloff1, F Hossner, M Voyle, J Ranson, J Powles, G Riley, G Sanger.   

Abstract

Three metabolites of N-[(1-butyl-4-piperidinyl)methyl]-3,4-dihydro-2H-[1,3]-oxazino[3,2_a]indole-10-carboxamide (SB-207266) (1) were synthesised and their pharmacological activity determined.

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Year:  2001        PMID： 11504648     DOI： 10.1016/s0968-0896(01)00120-1

Source DB:  PubMed          Journal:  Bioorg Med Chem        ISSN： 0968-0896            Impact factor:   3.641


  3 in total

1.  6,9-Dimeth-oxy-3,4-dihydro-1H-1,4-oxazino[4,3-a]indol-1-one.

Authors:  Cristian O Salas; Ricardo A Tapia; Yolanda Prieto
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2011-01-12

2.  A new host cell internalisation pathway for SadA-expressing staphylococci triggered by excreted neurochemicals.

Authors:  Arif Luqman; Patrick Ebner; Sebastian Reichert; Peter Sass; Clement Kabagema-Bilan; Christine Heilmann; Peter Ruth; Friedrich Götz
Journal:  Cell Microbiol       Date:  2019-06-07       Impact factor: 3.715

3.  Monoindole alkaloids from a marine sponge Spongosorites sp.

Authors:  Baoquan Bao; Ping Zhang; Yoonmi Lee; Jongki Hong; Chong-O Lee; Jee H Jung
Journal:  Mar Drugs       Date:  2007-06-25       Impact factor: 5.118
  3 in total

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