Literature DB >> 11501157

Triptolide: a potent inhibitor of NF-kappa B in T-lymphocytes.

H Liu1, Z H Liu, Z H Chen, J W Yang, L S Li.   

Abstract

AIM: To study the effect of triptolide on the activity of nuclear factor-kappa B (NF-kappa B) and gene expression of I kappa B alpha, a major inhibitor of NF-kappa B, in human Jurkat T cell line.
METHODS: Jurkat cells treated with or without PMA/PHA were incubated with varied doses of triptolide for different time periods. The activity of NF-kappa B in Jurkat cells was measured with electrophoretic mobility shift assays (EMSA), and the mRNA expression of I kappa B alpha in Jurkat cells was detected by semi-quantitative reverse transcription-polymerase chain reaction (RT-PCR).
RESULTS: PMA/PHA treatment was found to induce NF-kappa B activation rapidly. Triptolide treatment decreased the activity of NF-kappa B in both PMA/PHA treated and untreated Jurkat cells. This effect of triptolide was in a dose-dependent manner and was more obvious in cells treated with PMA/PHA. The mRNA expression of I kappa B alpha were upregulated by triptolide, while this effect was more potent in cells without PMA/PHA treatment.
CONCLUSION: Triptolide is a potent inhibitor of NF-kappa B activation in T lymphocyte and this effect is partly due to the upregulation of I kappa B alpha mRNA expression.

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Year:  2000        PMID: 11501157

Source DB:  PubMed          Journal:  Acta Pharmacol Sin        ISSN: 1671-4083            Impact factor:   6.150


  18 in total

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2.  Correspondence.

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3.  Triptolide-Assisted Phosphorylation of p53 Suppresses Inflammation-Induced NF-κB Survival Pathways in Cancer Cells.

Authors:  Li Zheng; Jia Jia; Huifang Dai; Lei Wan; Jian Liu; Lin Hu; Mian Zhou; Michael Qiu; Xufeng Chen; Lufen Chang; Jae Y Kim; Karen Reckamp; Dan J Raz; Zongping Xia; Binghui Shen
Journal:  Mol Cell Biol       Date:  2017-07-14       Impact factor: 4.272

4.  Triptolide, a constituent of immunosuppressive Chinese herbal medicine, is a potent suppressor of dendritic-cell maturation and trafficking.

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Review 5.  Drug discovery for polycystic kidney disease.

Authors:  Ying Sun; Hong Zhou; Bao-xue Yang
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Review 6.  A Chinese herb Tripterygium wilfordii Hook F in the treatment of rheumatoid arthritis: mechanism, efficacy, and safety.

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7.  GD3 synthase regulates epithelial-mesenchymal transition and metastasis in breast cancer.

Authors:  T R Sarkar; V L Battula; S J Werden; G V Vijay; E Q Ramirez-Peña; J H Taube; J T Chang; N Miura; W Porter; N Sphyris; M Andreeff; S A Mani
Journal:  Oncogene       Date:  2014-08-11       Impact factor: 9.867

8.  Triptolide-induced suppression of phospholipase D expression inhibits proliferation of MDA-MB-231 breast cancer cells.

Authors:  Dong Woo Kang; Ji Young Lee; Deuk Hee Oh; Seon Yang Park; Tae Min Woo; Mi Kyoung Kim; Mi Hee Park; Young Hoon Jang; Do Sik Min
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9.  Triptolide is a traditional Chinese medicine-derived inhibitor of polycystic kidney disease.

Authors:  Stephanie J Leuenroth; Dayne Okuhara; Joseph D Shotwell; Glen S Markowitz; Zhiheng Yu; Stefan Somlo; Craig M Crews
Journal:  Proc Natl Acad Sci U S A       Date:  2007-03-06       Impact factor: 11.205

10.  Effects of triptolide from Radix Tripterygium wilfordii (Leigongteng) on cartilage cytokines and transcription factor NF-kappaB: a study on induced arthritis in rats.

Authors:  Cheng Xiao; Jing Zhou; Yinghui He; Hongwei Jia; Linhua Zhao; Ning Zhao; Aiping Lu
Journal:  Chin Med       Date:  2009-07-02       Impact factor: 5.455

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