Literature DB >> 11490303

Effects of isoproterenol and butylscopolamine on the friction between an artificial stone and the intraureteral wall in anesthetized rabbits.

R Miyatake1, Y Tomiyama, M Murakami, Y C Park, T Kurita.   

Abstract

PURPOSE: We evaluated the effects of the nonselective beta-adrenoceptor agonist isoproterenol and the nonselective muscarinic antagonist butylscopolamine on ureteral wall tension, namely friction between an artificial stone and the intraureteral wall, in anesthetized rabbits.
MATERIALS AND METHODS: The relaxing effect of the drugs on the KCl induced tonic contraction was examined in isolated rabbit ureters. The effect of the drugs on the applied force needed for the artificial stone to pass at a constant speed through the ureter, called sliding force, was evaluated in anesthetized rabbits.
RESULTS: In a concentration dependent manner isoproterenol but not butylscopolamine reduced the KCl induced contraction in isolated ureter (mean pD2 7.35 +/- 0.06). Intravenous administration of 1 and 10 microg./kg. isoproterenol significantly decreased the friction between the artificial stone and intraureteral wall in anesthetized rabbits with sliding force at 15 minutes after drug administration decreased by 54.5% and 63.6%, respectively. In contrast, 100 and 1,000 microg./kg. butylscopolamine intravenously had no evident effect on ureteral wall tension.
CONCLUSIONS: Our results strongly suggest that ureteral smooth muscle relaxation by beta-adrenergic stimulation reduces ureteral wall tension, thereby, diminishing mechanical effects impeding the movement of a ureteral stone down the ureter.

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Year:  2001        PMID: 11490303

Source DB:  PubMed          Journal:  J Urol        ISSN: 0022-5347            Impact factor:   7.450


  3 in total

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Journal:  Can Urol Assoc J       Date:  2014 Jan-Feb       Impact factor: 1.862

2.  The potency of KUL-7211, a selective ureteral relaxant, in isolated canine ureter: comparison with various spasmolytics.

Authors:  Isao Wanajo; Yoshitaka Tomiyama; Mariko Tadachi; Mamoru Kobayashi; Yoshinobu Yamazaki; Masami Kojima; Nobuo Shibata
Journal:  Urol Res       Date:  2005-08-25

3.  Does the use of doxazosin influence the success of SWL in the treatment of upper ureteral stones? A multicenter, prospective and randomized study.

Authors:  Ferhat Ateş; Bilal Eryıldırım; Metin Ishak Öztürk; Turgay Turan; Cenk Gürbüz; Mete Oğuz Ekinci; Asıf Yıldırım; Cemal Göktaş; Temuçin Şenkul; Kemal Sarıca
Journal:  Urol Res       Date:  2012-01-07
  3 in total

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