Literature DB >> 11465425

Microhardness and dislocation identification studies on paracetamol single crystals.

S Finnie1, K V Prasad, D B Sheen, J N Sherwood.   

Abstract

PURPOSE: To study the mechanical behaviour of paracetamol single crystals.
METHODS: Microhardness indentation techniques were used to study the hardness anisotropy of paracetamol. Solvent etching technique was used to define the range of plastic deformation and the orientation of the dislocation lines. The orientation dependence of Knoop hardness on the (001), (110) and (201) surfaces was compared with calculated values of the Effective Resolved Shear Stress (ERSS) for plastic deformation by specific dislocation types.
RESULTS: The principal habit faces of single crystals using both Vickers and Knoop indenters showed a range of hardness from 235 to 456 MPa depending on the type of indenter used and its orientation on the surface. Solvent etching of the plastically deformed region of the crystal around the Vickers/Knoop indentations confirmed that the slip plane was (010). ERSS analysis suggested that the deformation occurred by the slip of dislocations of the types (010)[001] and (010)[100]. Crystals doped with 0.08-0.8 w/w% p-acetoxyacetanilide showed hardness values similar to the pure material.
CONCLUSIONS: The low number of distinct dislocation slip systems (two) is characteristic of a brittle material and is consistent with the observation that paracetamol will tolerate only deformations of 1 part in 10(6) before fracture.

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Year:  2001        PMID: 11465425     DOI: 10.1023/a:1011093612868

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  6 in total

1.  Fracture property studies of paracetamol single crystals using microindentation techniques.

Authors:  K V Prasad; D B Sheen; J N Sherwood
Journal:  Pharm Res       Date:  2001-06       Impact factor: 4.200

2.  Topochemistry of the initial stages of the dissolution of single crystals of acetaminophen.

Authors:  M A Vasil'chenko; T P Shakhtshneider; V V Boldyrev
Journal:  J Pharm Sci       Date:  1996-09       Impact factor: 3.534

3.  The effect of crystal hardness on compaction propensity.

Authors:  J Ichikawa; K Imagawa; N Kaneniwa
Journal:  Chem Pharm Bull (Tokyo)       Date:  1988-07       Impact factor: 1.645

4.  Unloading and postcompression viscoelastic stress versus strain behavior of pharmaceutical solids.

Authors:  D W Danielson; W T Morehead; E G Rippie
Journal:  J Pharm Sci       Date:  1983-04       Impact factor: 3.534

5.  Crystallization of paracetamol from solution in the presence and absence of impurity.

Authors:  K V Prasad; R I Ristic; D B Sheen; J N Sherwood
Journal:  Int J Pharm       Date:  2001-03-14       Impact factor: 5.875

6.  Hardness anisotropy of acetaminophen crystals.

Authors:  W C Duncan-Hewitt; D L Mount; A Yu
Journal:  Pharm Res       Date:  1994-05       Impact factor: 4.200

  6 in total
  4 in total

1.  Overcoming poor tabletability of pharmaceutical crystals by surface modification.

Authors:  Limin Shi; Changquan Calvin Sun
Journal:  Pharm Res       Date:  2011-06-28       Impact factor: 4.200

2.  Fracture property studies of paracetamol single crystals using microindentation techniques.

Authors:  K V Prasad; D B Sheen; J N Sherwood
Journal:  Pharm Res       Date:  2001-06       Impact factor: 4.200

3.  Mechanical properties of β-HMX.

Authors:  Hugh G Gallagher; John C Miller; David B Sheen; John N Sherwood; Ranko M Vrcelj
Journal:  Chem Cent J       Date:  2015-04-18       Impact factor: 4.215

4.  Growth and dislocation studies of β-HMX.

Authors:  Hugh G Gallagher; John N Sherwood; Ranko M Vrcelj
Journal:  Chem Cent J       Date:  2014-12-19       Impact factor: 4.215

  4 in total

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