Literature DB >> 11451044

Profound effect of plasma protein binding on the polarized transport of furosemide and verapamil in the Caco-2 model.

S M Chung1, E J Park, S M Swanson, T C Wu, W L Chiou.   

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Year:  2001        PMID: 11451044     DOI: 10.1023/a:1011022931368

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


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  22 in total

1.  Evaluation of an accelerated Caco-2 cell permeability model.

Authors:  E Liang; K Chessic; M Yazdanian
Journal:  J Pharm Sci       Date:  2000-03       Impact factor: 3.534

2.  Link between drug absorption solubility and permeability measurements in Caco-2 cells.

Authors:  V Pade; S Stavchansky
Journal:  J Pharm Sci       Date:  1998-12       Impact factor: 3.534

Review 3.  Intestinal drug absorption and metabolism in cell cultures: Caco-2 and beyond.

Authors:  P Artursson; R T Borchardt
Journal:  Pharm Res       Date:  1997-12       Impact factor: 4.200

4.  Persistent inhibition of CYP3A4 by ketoconazole in modified Caco-2 cells.

Authors:  M A Gibbs; M T Baillie; D D Shen; K L Kunze; K E Thummel
Journal:  Pharm Res       Date:  2000-03       Impact factor: 4.200

5.  Pharmacokinetics and pharmacodynamics of high dose furosemide in patients with chronic renal failure or nephrotic syndrome.

Authors:  H J Kühnel; K Günther; G Stein; A Hoffmann-Traeger
Journal:  Int J Clin Pharmacol Ther Toxicol       Date:  1987-11

6.  Influence of P-glycoprotein on the transport and metabolism of indinavir in Caco-2 cells expressing cytochrome P-450 3A4.

Authors:  J H Hochman; M Chiba; J Nishime; M Yamazaki; J H Lin
Journal:  J Pharmacol Exp Ther       Date:  2000-01       Impact factor: 4.030

7.  Characterization of the regional intestinal kinetics of drug efflux in rat and human intestine and in Caco-2 cells.

Authors:  V D Makhey; A Guo; D A Norris; P Hu; J Yan; P J Sinko
Journal:  Pharm Res       Date:  1998-08       Impact factor: 4.200

8.  Evaluation of potential causes for the incomplete bioavailability of furosemide: gastric first-pass metabolism.

Authors:  M G Lee; W L Chiou
Journal:  J Pharmacokinet Biopharm       Date:  1983-12

9.  Intravenous verapamil kinetics in rats: marked arteriovenous concentration difference and comparison with humans.

Authors:  P Manitpisitkul; W L Chiou
Journal:  Biopharm Drug Dispos       Date:  1993-10       Impact factor: 1.627

10.  Binding of phenothiazine neuroleptics to plasma proteins.

Authors:  R K Verbeeck; J A Cardinal; A G Hill; K K Midha
Journal:  Biochem Pharmacol       Date:  1983-09-01       Impact factor: 5.858

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  3 in total

Review 1.  Theoretical predictions of drug absorption in drug discovery and development.

Authors:  Patric Stenberg; Christel A S Bergström; Kristina Luthman; Per Artursson
Journal:  Clin Pharmacokinet       Date:  2002       Impact factor: 6.447

2.  Using Human Plasma as an Assay Medium in Caco-2 Studies Improves Mass Balance for Lipophilic Compounds.

Authors:  Kasiram Katneni; Thao Pham; Jessica Saunders; Gong Chen; Rahul Patil; Karen L White; Nada Abla; Francis C K Chiu; David M Shackleford; Susan A Charman
Journal:  Pharm Res       Date:  2018-09-17       Impact factor: 4.200

Review 3.  Fitting Transporter Activities to Cellular Drug Concentrations and Fluxes: Why the Bumblebee Can Fly.

Authors:  Pedro Mendes; Stephen G Oliver; Douglas B Kell
Journal:  Trends Pharmacol Sci       Date:  2015-11-01       Impact factor: 14.819

  3 in total

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