Literature DB >> 11440589

N-(tert-butoxycarbonyl)-N-[4-(dimethylazaniumylidene)-1,4-dihydropyridin-1-ylsulfonyl]azanide: a new sulfamyolating agent. Structure and reactivity toward amines.

J Y Winum1, L Toupet, V Barragan, G Dewynter, J L Montero.   

Abstract

[structure: see text] Synthesis, structure, and reactivity toward amines of the new sulfamoylating reagent 2 are described. Compound 2 allowed sulfamoylation of amines under very mild conditions to give sulfamide derivatives in good yields.

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Year:  2001        PMID： 11440589     DOI： 10.1021/ol0161312

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  7 in total

1.  Synthesis of chromone, quinolone, and benzoxazinone sulfonamide nucleosides as conformationally constrained inhibitors of adenylating enzymes required for siderophore biosynthesis.

Authors:  Curtis A Engelhart; Courtney C Aldrich
Journal:  J Org Chem       Date:  2013-07-12       Impact factor: 4.354

2.  Photochemically Mediated Nickel-Catalyzed Synthesis of N-(Hetero)aryl Sulfamides.

Authors:  R Thomas Simons; Georgia E Scott; Anastasia Gant Kanegusuku; Jennifer L Roizen
Journal:  J Org Chem       Date:  2020-05-04       Impact factor: 4.354

3.  Alternative method of Boc-removal from sulfamide using silica-phenyl sulfonic acid in conjunction with microwave heating.

Authors:  Shahnaz Ghassemi; Kristin Fuchs
Journal:  Mol Divers       Date:  2005       Impact factor: 2.943

4.  Discovery and Pharmacokinetics of Sulfamides and Guanidines as Potent Human Arginase 1 Inhibitors.

Authors:  Roman Blaszczyk; Joanna Brzezinska; Barbara Dymek; Paulina S Stanczak; Marcin Mazurkiewicz; Jacek Olczak; Julita Nowicka; Karolina Dzwonek; Agnieszka Zagozdzon; Jakub Golab; Adam Golebiowski
Journal:  ACS Med Chem Lett       Date:  2020-03-13       Impact factor: 4.345

5.  Discovery of spiro-piperidine inhibitors and their modulation of the dynamics of the M2 proton channel from influenza A virus.

Authors:  Jun Wang; Sarah D Cady; Victoria Balannik; Lawrence H Pinto; William F DeGrado; Mei Hong
Journal:  J Am Chem Soc       Date:  2009-06-17       Impact factor: 15.419

6.  Identification of novel pyrrolopyrimidine and pyrrolopyridine derivatives as potent ENPP1 inhibitors.

Authors:  Hee Jin Jeong; Hye Lim Lee; Sung Joon Kim; Jeong Hyun Jeong; Su Hyun Ji; Han Byeol Kim; Miso Kang; Hwan Won Chung; Chan Sun Park; Hyunah Choo; Hyo Jae Yoon; Nam-Jung Kim; Duck-Hyung Lee; Sang Hee Lee; Seo-Jung Han
Journal:  J Enzyme Inhib Med Chem       Date:  2022-12       Impact factor: 5.756

7.  Synthesis, Antiproliferative Activity and Molecular Docking Studies of Novel Doubly Modified Colchicine Amides and Sulfonamides as Anticancer Agents.

Authors:  Julia Krzywik; Witold Mozga; Maral Aminpour; Jan Janczak; Ewa Maj; Joanna Wietrzyk; Jack A Tuszyński; Adam Huczyński
Journal:  Molecules       Date:  2020-04-14       Impact factor: 4.411
  7 in total

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