Literature DB >> 11354357

Two novel and potent 3-[(o-methoxyphenyl)piperazinylethyl]-5-phenylthien.

W A Carroll1, K B Sippy, T A Esbenshade, S A Buckner, A A Hancock, M D Meyer.   

Abstract

The synthesis and in vitro characterization of A-119637 and A-123189, two novel, selective and potent alpha1D antagonists, are described.

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Year:  2001        PMID： 11354357     DOI： 10.1016/s0960-894x(01)00159-7

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

1.  The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptors.

Authors:  Stephen P H Alexander; Helen E Benson; Elena Faccenda; Adam J Pawson; Joanna L Sharman; Michael Spedding; John A Peters; Anthony J Harmar
Journal:  Br J Pharmacol       Date:  2013-12       Impact factor: 8.739

Review 2.  Adrenergic control of cardiac gap junction function and expression.

Authors:  Aida Salameh; Stefan Dhein
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2011-02-12       Impact factor: 3.000

3.  Involvement of the α(1D)-adrenergic receptor in methamphetamine-induced hyperthermia and neurotoxicity in rats.

Authors:  Kazue Kikuchi-Utsumi; Mami Ishizaka; Nobuko Matsumura; Masahiko Watabe; Koji Aoyama; Nobuyuki Sasakawa; Toshio Nakaki
Journal:  Neurotox Res       Date:  2013-01-03       Impact factor: 3.911

4.  Smooth muscle alpha1D-adrenoceptors mediate phenylephrine-induced vasoconstriction and increases in endothelial cell Ca2+ in hamster cremaster arterioles.

Authors:  W F Jackson; E M Boerman; E J Lange; S S Lundback; K D Cohen
Journal:  Br J Pharmacol       Date:  2008-07-07       Impact factor: 8.739

5.  Enhancement of apomorphine-induced penile erection in the rat by a selective alpha(1D)-adrenoceptor antagonist.

Authors:  Hiroya Mizusawa; Petter Hedlund; Johan Sjunnesson; Jorge D Brioni; James P Sullivan; Karl-Erik Andersson
Journal:  Br J Pharmacol       Date:  2002-07       Impact factor: 8.739

6.  Alpha-1-adrenoceptor subtype selective regulation of connexin 43 expression in rat cardiomyocytes.

Authors:  Diana Marcela Rojas Gomez; Jan Sebastian Schulte; Friedrich-Wilhelm Mohr; Stefan Dhein
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  2008-01-08       Impact factor: 3.000
  6 in total

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