Literature DB >> 11318765

Lack of effect of ondansetron on the pharmacokinetics and analgesic effects of morphine and metabolites after single-dose morphine administration in healthy volunteers.

K R Crews1, B P Murthy, E K Hussey, A N Passannante, J L Palmer, W Maixner, K L Brouwer.   

Abstract

AIMS: The purpose of this investigation was to study the influence of ondansetron on the single-dose pharmacokinetics and the analgesic effects elicited by morphine and the 3- and 6-glucuronide metabolites of morphine in healthy volunteers.
METHODS: This was a randomized, double-blind, placebo-controlled, two-way crossover study in which six male and six female subjects were administered a single 10 mg intravenous dose of morphine sulphate, followed 30 min later by a single 16 mg intravenous dose of ondansetron hydrochloride or placebo. Serum and urine concentrations of morphine, morphine-3-glucuronide (M3G) and morphine-6-glucuronide (M6G) samples were quantified over 48 h using high performance liquid chromatography with detection by mass spectrometry. Analgesia was assessed in the volunteers with a contact thermode device to provide a thermal pain stimulus. Four analgesic response variables were measured including thermal pain threshold, thermal pain tolerance, temporal summation of pain and mood state.
RESULTS: The two treatments appeared to be equivalent based on the 90% confidence intervals (0.6, 1.67) of the least squares means ratio. All least squares means ratio confidence intervals for each parameter, for each analyte fell within the specified range, demonstrating a lack of an interaction.
CONCLUSIONS: The results of this study suggest that administration of ondansetron (16 mg i.v.) does not alter the pharmacokinetics of morphine and its 3- or 6-glucuronide metabolites to a clinically significant extent, nor does it affect the overall analgesic response to morphine as measured by the contact thermode system.

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Year:  2001        PMID: 11318765      PMCID: PMC2014461          DOI: 10.1046/j.1365-2125.2001.01369.x

Source DB:  PubMed          Journal:  Br J Clin Pharmacol        ISSN: 0306-5251            Impact factor:   4.335


  13 in total

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Authors:  G M Pacifici; A Rane
Journal:  Drug Metab Dispos       Date:  1981 Nov-Dec       Impact factor: 3.922

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Authors:  W Maixner; R Fillingim; A Sigurdsson; S Kincaid; S Silva
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Review 8.  Pain and the placebo response.

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9.  Probenecid impairment of acetaminophen and lorazepam clearance: direct inhibition of ether glucuronide formation.

Authors:  D R Abernethy; D J Greenblatt; B Ameer; R I Shader
Journal:  J Pharmacol Exp Ther       Date:  1985-08       Impact factor: 4.030

10.  A psychophysical analysis of morphine analgesia.

Authors:  D D Price; A Von der Gruen; J Miller; A Rafii; C Price
Journal:  Pain       Date:  1985-07       Impact factor: 6.961

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