E A Sudbeck1, S Ghosh, X P Liu, Y Zheng, D E Myers, F M Uckun. Show Affiliations » 1. Parker Hughes Cancer Center and Drug Discovery Program, Parker Hughes Institute, St. Paul, MN, USA.
Abstract
Entities: Disease
Mesh: See more » Adenocarcinoma/pathologyAmides/chemistryAmides/pharmacologyAmides/therapeutic useAniline Compounds/chemical synthesisAniline Compounds/chemistryAniline Compounds/pharmacologyAniline Compounds/therapeutic useAnimalsAntineoplastic Agents/chemistryAntineoplastic Agents/pharmacologyAntineoplastic Agents/therapeutic useAntineoplastic Agents/toxicityBreast Neoplasms/pathologyDrug DesignEnzyme Inhibitors/chemistryEnzyme Inhibitors/pharmacologyEnzyme Inhibitors/therapeutic useEpidermal Growth Factor/chemistryEpidermal Growth Factor/pharmacologyEpidermal Growth Factor/therapeutic useEpidermal Growth Factor/toxicityErbB Receptors/antagonists & inhibitorsErbB Receptors/chemistryErbB Receptors/drug effectsFemaleGenistein/chemistryGenistein/pharmacologyGenistein/therapeutic useGenistein/toxicityHumansLeukemia/drug therapyLeukemia/pathologyMacaca fascicularisMiceMice, Inbred BALB CMice, SCIDModels, MolecularMolecular StructureNeoplasm Proteins/antagonists & inhibitorsNeoplasm Proteins/chemistryNeoplasm Proteins/drug effectsNeoplasms/drug therapyNeoplasms/enzymologyNitriles/chemical synthesisNitriles/chemistryNitriles/pharmacologyNitriles/therapeutic useProtein ConformationProtein Structure, TertiaryQuinazolines/chemical synthesisQuinazolines/chemistryQuinazolines/pharmacologyQuinazolines/therapeutic useRecombinant Fusion Proteins/antagonists & inhibitorsSequence AlignmentSpecies SpecificityStructure-Activity RelationshipTumor Cells, Cultured/drug effectsTumor Stem Cell AssayXenograft Model Antitumor Assays
Substances: See more » AmidesAniline CompoundsAntineoplastic AgentsEGF-genisteinEnzyme InhibitorsLFM A12LFM A13Neoplasm ProteinsNitrilesQuinazolinesRecombinant Fusion ProteinsWHI P154WHI P97Epidermal Growth FactorGenisteinErbB Receptors
Year: 2001 PMID: 11217368 DOI: 10.1385/1-59259-114-0:193
Source DB: PubMed Journal: Methods Mol Biol ISSN: 1064-3745