Literature DB >> 11150162

Design and synthesis of new orally active nonpeptidic inhibitors of human neutrophil elastase.

K Ohmoto1, T Yamamoto, T Horiuchi, H Imanishi, Y Odagaki, K Kawabata, T Sekioka, Y Hirota, S Matsuoka, H Nakai, M Toda, J C Cheronis, L W Spruce, A Gyorkos, M Wieczorek.   

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Year:  2000        PMID： 11150162     DOI： 10.1021/jm0004087

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  4 in total

1.  Synthesis, X-ray diffraction analysis, quantum chemical studies and α-amylase inhibition of probenecid derived S-alkylphthalimide-oxadiazole-benzenesulfonamide hybrids.

Authors:  Bilal Ahmad Khan; Syeda Shamila Hamdani; Muhammad Naeem Ahmed; Shahid Hameed; Muhammad Ashfaq; Ahmed M Shawky; Mahmoud A A Ibrahim; Peter A Sidhom
Journal:  J Enzyme Inhib Med Chem       Date:  2022-12       Impact factor: 5.756

Review 2.  Emerging challenges in the design of selective substrates, inhibitors and activity-based probes for indistinguishable proteases.

Authors:  Paulina Kasperkiewicz; Marcin Poreba; Katarzyna Groborz; Marcin Drag
Journal:  FEBS J       Date:  2017-01-29       Impact factor: 5.542

3.  Synthesis and biological evaluation of dehydroabietic acid-pyrimidine hybrids as antitumor agents.

Authors:  Lin Huang; Rong Huang; Fuhua Pang; Anke Li; Guobao Huang; Xiaoqun Zhou; Qian Li; Fangyao Li; Xianli Ma
Journal:  RSC Adv       Date:  2020-05-11       Impact factor: 4.036

Review 4.  Synthetic approaches and pharmacological activity of 1,3,4-oxadiazoles: a review of the literature from 2000-2012.

Authors:  Cledualdo Soares de Oliveira; Bruno Freitas Lira; José Maria Barbosa-Filho; Jorge Gonçalo Fernandez Lorenzo; Petrônio Filgueiras de Athayde-Filho
Journal:  Molecules       Date:  2012-08-27       Impact factor: 4.411
  4 in total

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